Search Result "inhibitor"


Mini-Review Article

Approach in Improving Potency and Selectivity of Kinase Inhibitors: Allosteric Kinase Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 21 Issue: 8 Year: 2021 Page: 991-1003
Author(s): Shangfei Wei,Tianming Zhao,Jie Wang,Xin Zhai

Review Article

Monoclonal Antibodies, Small Molecule Inhibitors and Antibody-drug Conjugates as HER2 Inhibitors

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 1 Year: 2021 Page: 3339-3360
Author(s): Xiu-Fang Li,Chen-Fu Liu,Guo-Wu Rao

Review Article

Is It the Twilight of BACE1 Inhibitors?

Journal: Current Neuropharmacology
Volume: 19 Issue: 1 Year: 2021 Page: 61-77
Author(s): Martina Hrabinova,Jaroslav Pejchal,Tomas Kucera,Daniel Jun,Monika Schmidt,Ondrej Soukup

Review Article

Relevance of Aromatase Inhibitors in Breast Cancer Treatment

Journal: Current Topics in Medicinal Chemistry
Volume: 21 Issue: 0 Year: 2021 Page: 1-18
Author(s): Ankita Sood,Damanpreet Kaur Lang,Rajwinder Kaur,Balraj Saini,Sandeep Arora

Review Article

Current Status of SUMOylation Inhibitors

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 2 Year: 2021 Page: 3892-3912
Author(s): Christopher M. Brackett,Brian S.J. Blagg

Review Article

Efficacy and cardiovascular safety of SGLT2 Inhibitors

Journal: Current Drug Safety
Volume: 16 Issue: 2 Year: 2021 Page: 178-196
Author(s): Cornelius James Fernandez,Abisha Graciano Nevins,Shasta Nawaz,Tahir Nazir,Fahmy W F Hanna

General Review Article

Janus Kinase Inhibitors: A Review of Their Application in the Vitiligo

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 21 Issue: 2 Year: 2021 Page: 3203-3218
Author(s): Chao Niu,Hunjun Xie,Haji Akber Aisa

Review Article

Recent Advances in the Development of Casein Kinase 1 Inhibitors

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 8 Year: 2021 Page: 1585-1604
Author(s): Sha-Sha Li,Yue-Hui Dong,Zhao-Peng Liu

Review Article

The Effect of PDE5 Inhibitors on the Male Reproductive Tract

Journal: Current Pharmaceutical Design
Volume: 27 Issue: 2 Year: 2021 Page: 2697-2713
Author(s): Nikolaos Sofikitis,Aris Kaltsas,Fotios Dimitriadis,Jens Rassweiler,Nikolaos Grivas,Athanasios Zachariou,Apostolos Kaponis,Panagiota Tsounapi,Napoleon Paterakis,Andreas Karagiannis,Sotirios Skouros,Ioannis Giannakis,Ioannis Champilomatis,Minas Paschopoulos,Diamantis Daphnis,Ioannis Giakoumakis,Melinda R.Gabales,Jo Ben M. Chua,Pedro L. Lantin III,Charalampos Mamoulakis,Atsushi Takenaka

Mini-Review Article

Recent Progress on the Discovery of NLRP3 Inhibitors and their Therapeutic Potential

Journal: Current Medicinal Chemistry
Volume: 28 Issue: 3 Year: 2021 Page: 569-582
Author(s): Ma Su,Weiwei Wang,Feng Liu,Huanqiu Li

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