Search Result "in vitro potency"


Influence of Polymer Molecular Weight on in-vitro Characteristics and Cytotoxicity of Fulvestrant Loaded Nanoparticles

Journal: Current Drug Therapy
Volume: 9 Issue: 4 Year: 2014 Page: 239-249
Author(s): Canan Hascicek,Ceyda T. Sengel-Turk,Mehmet Gumustas,Sibel A. Ozkan,Filiz Bakar,Net Das-Evcimen,Ayhan Savaser,Yalcin Ozkan

Knocking on FXR's Door:The Hammerhead-Structure Series of FXRs Agonists - Amphiphilic Isoxazoles with Potent In Vitro and In Vivo Activities

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 19 Year: 2014 Page: 2143-2158
Author(s): Christian Gege,Olaf Kinzel,Christoph Steeneck,Andreas Schulz,Claus Kremoser

Microbiological Assay for the Determination of Colistin Sulphate

Journal: Current Analytical Chemistry
Volume: 10 Issue: 3 Year: 2014 Page: 443-448
Author(s): Giovana Calixto, Luciana Elisete Domingos, Nathalie Thomazini Fabri, Thais Adriana do Carmo, Andreia de Haro Moreno, Herida Regina Nunes Salgado, Marlus Chorilli

Synthesis and In Vitro Evaluation of Novel 1,2,3,4-Tetrahydroisoquinoline Derivatives as Potent Antiglioma Agents

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 14 Issue: 3 Year: 2014 Page: 473-482
Author(s): Renukadevi Patil,Amira Hosni-Ahmed,Terreia S. Jones,Shivaputra A. Patil,Likeselam B. Asres,Xiangdi Wang,Ryan C. Yates,Eldon E. Geisert,Duane D. Miller

Synthesis, Molecular Docking and In Vitro Antimicrobial Studies of Novel Pyrazole Analogues of Curcumin

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 4 Year: 2014 Page: 474-483
Author(s): Dileep Kumar,Harish B. G.,Mayank Gangwar,Manish Kumar,Dharmendra Kumar,Ragini Tilak,Gopal Nath,Ashok Kumar,Sushil Kumar Singh

In Vitro and In Vivo Activities of Novel Cyclic Lipopeptides Against Staphylococcal Biofilms

Journal: Protein & Peptide Letters
Volume: 21 Issue: 4 Year: 2014 Page: 352-356
Author(s): Nina Bionda,Irena Pastar,Stephen C. Davis,Predrag Cudic

Fluorinated Compounds in Medicinal Chemistry: Recent Applications, Synthetic Advances and Matched-Pair Analyses

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 7 Year: 2014 Page: 855-864
Author(s): David Barnes-Seeman,Jeremy Beck,Clayton Springer

In Vitro, In Vivo and In Silico Analysis of the Anticancer and Estrogen-like Activity of Guava Leaf Extracts

Journal: Current Medicinal Chemistry
Volume: 21 Issue: 20 Year: 2014 Page: 2322-2330
Author(s): L.Y. Rizzo,G.B. Longato,A.LT.G. Ruiz,S.V. Tinti,A. Possenti,D.B. Vendramini-Costa,A. Sartoratto,G.M. Figueira,F.L.N. Silva,M.N. Eberlin,T.A.C.B. Souza,M.T. Murakami,E. Rizzo,M.A. Foglio,F. Kiessling,T. Lammers,J.E. Carvalho

Synthesis of Novel 2,3,4-trisubstituted-oxazolidine Derivatives and In Vitro Cytotoxic Evaluation

Journal: Medicinal Chemistry
Volume: 10 Issue: 6 Year: 2014 Page: 609-618
Author(s): Saulo F. Andrad, Edmar F.S. Campos, Claudia S. Teixeira, Cristiano C. Bandeira, Stefania N. Lavorato, Nelilma C. Romeiro, Caryne M. Bertollo, Monica C. Oliveira, Elaine M. Souza-Fagundes, Ricardo J. Alves

Research Article

Steroidal Cardiac Na+/K+ ATPase Inhibitors Exhibit Strong Anti-Cancer Potential in vitro and in Prostate and Lung Cancer Xenografts in vivo

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 14 Issue: 5 Year: 2014 Page: 762-770
Author(s): Konstantinos Dimas, Natalia Papadopoulou, Constantinos Baskakis, Kyriakos C. Prousis, Michail Tsakos, Saad Alkahtani, Sabina Honisch, Florian Lang, Theodora Calogeropoulou, Konstantinos Alevizopoulos, Christos Stournaras

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