Search Result "hybrid pharmacophore approach"


Research Article

Design and Synthesis of 2-(Arylmethylideneamino) Isoindolines as New Potential Analgesic and Anti-Inflammatory Agents: A Molecular Hybridization Approach

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 37 Year: 2016 Page: 5760-5766
Author(s): Maryam Iman,Hamed Shafaroodi,Asghar Davood,Masoud Abedini,Pouyan Pishva,Mehrnoush Taherkhani,Ahmad Reza Dehpour,Abbas Shafiee

Design, Synthesis and Docking Study of Some Novel Isatin- Quinoline Hybrids as Potential Antitubercular Agents

Journal: Anti-Infective Agents
Volume: 14 Issue: 1 Year: 2016 Page: 53-62
Author(s): Srinubabu Maddela,Ajitha Makula

Research Article

Discovery of Camptothecin Based Topoisomerase I Inhibitors: Identification Using an Atom Based 3D-QSAR, Pharmacophore Modeling, Virtual Screening and Molecular Docking Approach

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 19 Issue: 9 Year: 2016 Page: 752-763
Author(s): Sanal Dev,Sunil R. Dhaneshwar,Bijo Mathew

In silico Studies Toward the Discovery of Novel Type-II Inhibitors of TrkA: Pharmacophore-based 3D-QSAR Modeling, Database Screening and Molecular Docking

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 6 Year: 2016 Page: 526-538
Author(s): Yahui Tian,Lu Zhou,Xiaoli Li,Suwen Zhou,Rong Yong,Liangliang Zhong

Review Article

Hybrid Bioactive Heterocycles as Potential Antimicrobial Agents: A Review

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2016 Page: 1500-1526
Author(s): Nisheeth Desai, Amit Trivedi, Unnat Pandit, Amit Dodiya, V. Kameswara Rao, Priyanka Desai

Systems Biology Approaches to a Rational Drug Discovery Paradigm

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 9 Year: 2016 Page: 1009-1025
Author(s): Philip Prathipati,Kenji Mizuguchi

Design and Synthesis of Novel Schiff Base-Benzothiazole Hybrids as Potential Epidermal Growth Factor Receptor (EGFR) Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 6 Year: 2016 Page: 722-739
Author(s): Meenakshi Singh,Sudhir Kumar Singh,Bhushan Thakur,Pritha Ray,Sushil K. Singh

Research Article

Novel Microwave Assisted Synthesis and Antimicrobial Activity of New Quinolone-Hybrids

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 9 Year: 2016 Page: 636-651
Author(s): Sule Ceylan,Hacer Bayrak,Serap Basoglu Ozdemir,Yıldız Uygun,Arif Mermer,Neslihan Demirbas,Serdar Ulker

Natural Products based P-glycoprotein Activators for Improved β-amyloid Clearance in Alzheimer’s Disease: An in silico Approach

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2016 Page: 50-59
Author(s): Pravin Shinde,Nikhil Vidyasagar,Sivakami Dhulap,Abhijeet Dhulap,Raj Hirwani

Review Article

Multitarget Opioid/Non-opioid Ligands: A Potential Approach in Pain Management

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 40 Year: 2016 Page: 4506-4528
Author(s): Rita Turnaturi,Giuseppina Arico,Giuseppe Ronsisvalle,Lorella Pasquinucci,Carmela Parenti

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