Search Result "fused pyrimidine"


Review Article

Pyrimidine-fused Derivatives: Synthetic Strategies and Medicinal Attributes

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 3175-3210
Author(s): Gaurav Joshi, Himanshu Nayyar, Jimi Marin Alex, Gajendra S. Vishwakarma, Sunil Mittal, Raj Kumar

Review Article

The Chemistry and Bio-Medicinal Significance of Pyrimidines & Condensed Pyrimidines

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 3133-3174
Author(s): K. S. Jain, N. Arya, N. N. Inamdar, P. B. Auti, S. A. Unawane, H. H. Puranik, M. S. Sanap, A. D. Inamke, V. J. Mahale, C. S. Prajapati, C. J. Shishoo

Research Article

Medicinal Chemistry Perspective of Fused Isoxazole Derivatives

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 2863-2883
Author(s): Mahesh A. Barmade, Prashant R. Murumkar, Mayank Kumar Sharma, Mange Ram Yadav

2, 7-Diarylidene-cycloheptanone, Hydrazonoyl Chlorides and Heterocyclic Amines as Precursors for Synthesis of Bioactive new Fused Cycloheptapyrimidine Derivatives

Journal: Current Organic Synthesis
Volume: 13 Issue: 2 Year: 2016 Page: 291-299
Author(s): Thoraya A. Farghaly,Magda A. Abdallah,Zeinab A. Muhammad

Cyclobutanones as Useful Synthons for the Preparation of Bioactive Molecules and Fused-Ring Chemicals

Journal: Current Organic Chemistry
Volume: 20 Issue: 1 Year: 2016 Page: 1878-1901
Author(s): Xiuyun Sun, Yonghui Sun, Yu Rao

Convergent Synthesis Strategy of Novel Fused Azines: 1H-15N HMBC NMR as a Tool for Assertion of the Site Selectivity of Aza-Michael Addition Reaction

Journal: Current Organic Synthesis
Volume: 13 Issue: 2 Year: 2016 Page: 278-290
Author(s): Tamer S. Saleh,Ahmed E. M. Mekky,Abdullah S. Al-Bogami

Research Article

Synthesis and In Vitro Activity of Pyrrolo[3,4-d]pyrimidine-2,5-diones as Potential Non-nucleoside HCV Inhibitors

Journal: Current Enzyme Inhibition
Volume: 12 Issue: 2 Year: 2016 Page: 170-176
Author(s): Amany S. Mostafa, Serry A. El Bialy, Waleed A. Bayoumi, Youki Ueda, Masanori Ikeda, Nobuyuki Kato, Ali M. Abdelal

Review Article

Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines and Structurally Simplified Analogs. Chemistry and SAR Profile as Adenosine Receptor Antagonists

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 3224-3257
Author(s): Sara Redenti, Antonella Ciancetta, Giorgia Pastorin, Barbara Cacciari, Stefano Moro, Giampiero Spalluto, Stephanie Federico

Investigation of the lactam-lactim and Thiolactam-thiolactim Tautomerism in the 2,2,5-Trimethylpyrano[4",3":4',5']pyrido[3',2':4,5]furo(thieno)[3,2-d]pyrimidines

Journal: Current Organic Chemistry
Volume: 20 Issue: 12 Year: 2016 Page: 1350-1358
Author(s): Samvel N. Sirakanyan,Domenico Spinelli,Athina Geronikaki,Henrik A. Panosyan,Anush A. Hovakimyan

Monocyclic and Fused Azines and Azoles as Histamine H4 Receptor Ligands

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 18 Year: 2016 Page: 1870-1925
Author(s): Dorota Lażewska,Enrique Domínguez-Álvarez,Katarzyna Kamińska,Kamil Kuder,Katarzyna Kieć-Kononowicz

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