Search Result "fragment discovery"


UCSF Small Molecule Discovery Center: Innovation, Collaboration and Chemical Biology in the Bay Area

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 17 Issue: 4 Year: 2014 Page: 333-342
Author(s): Michelle R. Arkin,Kenny K.H. Ang,Steven Chen,Julia Davies,Connie Merron,Yinyan Tang,Christopher G.M. Wilson,Adam R. Renslo

Molecular Imaging Aided Improvement in Drug Discovery and Development

Journal: Current Biotechnology
Volume: 3 Issue: 3 Year: 2014 Page: 218-237
Author(s): Smrita Chaudhury,Bhushan Thakur,Subhoshree Chatterjee,Pritha Ray

Impact of Computational Structure-based Methods on Drug Discovery

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 20 Year: 2014 Page: 3380-3386
Author(s): Charles H. Reynolds

Discovery of Novel Candidate Therapeutics and Diagnostics Based on Engineered Human Antibody Domains

Journal: Current Drug Discovery Technologies
Volume: 11 Issue: 1 Year: 2014 Page: 28-40
Author(s): Weizao Chen,Rui Gong,Tianlei Ying,Ponraj Prabakaran,Zhongyu Zhu,Yang Feng,Dimiter S. Dimitrov

Identifying Structural Features Related to the Biological Activity of a Series of AT1 Antagonists from Fragment-based Drug Design

Journal: Protein & Peptide Letters
Volume: 21 Issue: 6 Year: 2014 Page: 542-549
Author(s): Danielle da C. Silva,Vinícius G. Maltarollo,Kathia M. Honorio

From HTS to Phase I: The Institute for Therapeutics Discovery and Development at the University of Minnesota

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 17 Issue: 3 Year: 2014 Page: 231-240
Author(s): Peter I. Dosa,Gunda I. Georg,Vadim J. Gurvich,Jon E. Hawkinson,Michael A. Walters,Henry L. Wong

Multicomponent Reactions in Antimitotic Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 20 Year: 2014 Page: 2209-2230
Author(s): Angel Cores,Carlos Carbajales,Alberto Coelho

Methods for Docking Small Molecules to Macromolecules: A User’s Perspective. 2. Applications

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 20 Year: 2014 Page: 3360-3372
Author(s): Valerie Campagna-Slater,Eric Therrien,Nathanael Weill,Nicolas Moitessier

Biocomputational Resources Useful For Drug Discovery Against Compartmentalized Targets

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 2 Year: 2014 Page: 293-300
Author(s): Francisca Sanchez-Jimenez, Armando Reyes-Palomares, Aurelio A. Moya-Garcia, Juan AG Ranea, Miguel Angel Medina

Virtual Screening and Discovery of Novel Aurora Kinase Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 17 Year: 2014 Page: 2006-2019
Author(s): R. Raghu,Vinod Devaraji,K. Leena,Sd. Riyaz,Polavaru Baby Rani,Suneel Kumar. B,Pradeep Kumar Naik,P.K. Dubey,Devadasan Velmurugan,M. Vijayalakshmi

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