Search Result "efflux pump inhibitors"


Clinical Impact of the Over-Expression of Efflux Pump in Nonfermentative Gram-Negative Bacilli, Development of Efflux Pump Inhibitors

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 797-807
Author(s): Jordi Vila, Jose Luis Martinez

New Methods for the Identification of Efflux Mediated MDR Bacteria, Genetic Assessment of Regulators and Efflux Pump Constituents, Characterization of Efflux Systems and Screening for Inhibitors of Efflux Pumps

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 760-778
Author(s): M. Viveiros, M. Martins, I. Couto, L. Rodrigues, G. Spengler, A. Martins, J. E. Kristiansen, J. Molnar, L. Amaral

The AcrB Efflux Pump: Conformational Cycling and Peristalsis Lead to Multidrug Resistance

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 729-749
Author(s): Markus A. Seeger, Kay Diederichs, Thomas Eicher, Lorenz Brandstatter, Andre Schiefner, Francois Verrey, Klaas M. Pos

Promising Therapy of XDR-TB/MDR-TB with Thioridazine an Inhibitor of Bacterial Efflux Pumps

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 816-819
Author(s): L. Amaral, M. Martins, M. Viveiros, J. Molnar, J. E. Kristiansen

Membrane Permeability and Regulation of Drug “Influx and Efflux” in Enterobacterial Pathogens

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 750-759
Author(s): Anne Davin-Regli, Jean-Michel Bolla, Chloe E. James, Jean-Philippe Lavigne, Jacqueline Chevalier, Eric Garnotel, Alexander Molitor, Jean-Marie Pages

Biophysical Characterization of In- and Efflux in Gram-Negative Bacteria

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 789-796
Author(s): Helge Weingart, Mircea Petrescu, Mathias Winterhalter

2(3)-Aryl-thio(oxy)-methylquinoxaline Derivatives: A New Class of P-Glycoprotein-Mediated Drug Efflux Inhibitors

Journal: Medicinal Chemistry
Volume: 4 Issue: 3 Year: 2008 Page: 194-205
Author(s): Antonio Carta, Sandra Piras, Giuseppe Paglietti, Sabrina Pricl, Paolo La Colla, Bernardetta Busonera, Roberta Loddo

Enhanced Killing of Intracellular Pathogenic Bacteria by Phenothiazines and the Role of K+ Efflux Pumps of the Bacterium and the Killing Macrophage

Journal: Anti-Infective Agents in Medicinal Chemistry
Volume: 7 Issue: 1 Year: 2008 Page: 63-72
Author(s): L. Amaral, M. Martins, M. Viveiros

Inhibition of Efflux of Quinolines as New Therapeutic Strategy in Malaria

Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 7 Year: 2008 Page: 563-578
Author(s): Maud Henry, Sandrine Alibert, Christophe Rogier, Jacques Barbe, Bruno Pradines

Antimicrobial Resistance in Foodborne Pathogens - A Cause for Concern?

Journal: Current Drug Targets
Volume: 9 Issue: 9 Year: 2008 Page: 808-815
Author(s): Ciara Walsh, Seamus Fanning

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