Search Result "docking studies"


Review Article

Docking Studies for Multi-Target Drugs

Journal: Current Drug Targets
Volume: 18 Issue: 5 Year: 2017 Page: 592-604
Author(s): Luciana Scotti,Francisco J.B. Mendonca Junior,Hamilton M. Ishiki,Frederico F. Ribeiro,Rajeev K. Singla,Jose M. Barbosa Filho,Marcelo S. Da Silva,Marcus T. Scotti

Research Article

QSAR and Molecular Docking Studies on a Series of Cinnamic Acid Analogues as Epidermal Growth Factor Receptor (EGFR) Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 83-95
Author(s): Basheerulla Shaik,Omar Deeb,Vijay K. Agrawal,Satya P. Gupta

Research Article

Combined Approach of QSAR and Docking Studies for the Design of Local Anaesthetic Agents

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 3 Year: 2017 Page: 272-276
Author(s): Chunyan Zhang,Zhi Li,Jiahai Ma,Jing Zhang,Longming Zhang,Tao Li,Shijian Zheng

Research Article

Molecular Docking and Structure Activity Relationship Studies of NSAIDs. What do they Reveal about IC50?

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 8 Year: 2017 Page: 949-958
Author(s): Chrysoula Mikra,Georgios Rossos,Sotirios K. Hadjikakou,Nikolaos Kourkoumelis

Research Article

Molecular Docking and In Silico ADMET Study Reveals Flavonoids as a Potential Inhibitor of Aromatase

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 11 Year: 2017 Page: 1267-1276
Author(s): Umang Shah,Samir Patel,Mehul Patel,Jagat Upadhayay

Research Article

Docking and QSAR Studies of 1,4-Dihydropyridine Derivatives as Anti- Cancer Agent

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 12 Issue: 2 Year: 2017 Page: 174-185
Author(s): Shirin Mollazadeh, Jamal Shamsara, Maryam Iman, Farzin Hadizadeh

Research Article

Docking and QSAR Studies of Aryl-valproic Acid Derivatives to Identify Antiproliferative Agents Targeting the HDAC8

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 7 Year: 2017 Page: 927-940
Author(s): Heidy Martínez-Pacheco,Guillermo Ramírez-Galicia,Midalia Vergara-Arias,Jurg Gertsch,Jonathan Manuel Fragoso-Vazquez,David Mendez-Luna,A. L. Abujamra,Cabrera-Perez Laura Cristina,Rosales-Hernandez Martha Cecilia,I Mendoza-Lujambio,Jose Correa-Basurto

Research Article

Synthesis, Molecular Docking and Pharmacological Study of Pyrimidothiadiazinones and its bis-derivatives

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 4 Year: 2017 Page: 434-443
Author(s): Sobhi M. Gomha,Ikhlass M. Abbas,Mohamed A. A. Elneairy,Mahmoud M. Elaasser,Bazada K. A. Mabrouk

Research Article

Molecular Docking Studies of Novel Thiosemicarbazone-based Indoles as Potential PI3Kα Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 11 Year: 2017 Page: 1252-1258
Author(s): Dima A. Sabbah,Kamal Sweidan

Research Article

Docking-based 3D-QSAR Studies of Phosphodiesterase 9A Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 9 Year: 2017 Page: 986-998
Author(s): Changji Tan,Yinuo Wu,Yongxian Shao,Haibin Luo,Xuehua Zheng,Laiyou Wang

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