Search Result "cyclin-dependent kinase"


Quantum Mechanical Scoring: Structural and Energetic Insights into Cyclin-Dependent Kinase 2 Inhibition by Pyrazolo[1,5-a]pyrimidines

Journal: Current Computer-Aided Drug Design
Volume: 9 Issue: 1 Year: 2013 Page: 118-129
Author(s): Pathik S. Brahmkshatriya,Petr Dobes,Jindrich Fanfrlik,Jan Rezac,Kamil Paruch,Agnieszka Bronowska,Martin Lepsík,Pavel Hobza

PfRIO-2 Kinase is a Potential Therapeutic Target of Antimalarial Protein Kinase Inhibitors

Journal: Current Drug Discovery Technologies
Volume: 10 Issue: 1 Year: 2013 Page: 85-91
Author(s): Swagata Nag, KMN Prasad, Ananya Bhowmick, Rohitas Deshmukh, Vishal Trivedi

Kinase CK2 Inhibition: An Update

Journal: Current Medicinal Chemistry
Volume: 20 Issue: 5 Year: 2013 Page: 671-693
Author(s): G. Cozza, L. A. Pinna, S. Moro

Dual Inhibition of PI3-Kinase and mTOR in Renal Cell Carcinoma

Journal: Current Cancer Drug Targets
Volume: 13 Issue: 2 Year: 2013 Page: 126-142
Author(s): Daniel C. Cho, James W. Mier

Rational Approaches Towards Lead Optimization of Kinase Inhibitors: The Issue of Specificity

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 26 Year: 2013 Page: 4714-4738
Author(s): Preethi Badrinarayan,G. Narahari Sastry

Protein Phosphatase 2A as a Potential Target for Treatment of Adult T Cell Leukemia

Journal: Current Cancer Drug Targets
Volume: 13 Issue: 8 Year: 2013 Page: 829-842
Author(s): Naoki Mori,Chie Ishikawa,Jun-Nosuke Uchihara,Takeshi Yasumoto

Research Article

Gallic Acid Attenuates Oleic Acid-induced Proliferation of Vascular Smooth Muscle Cell Through Regulation of AMPK-eNOS-FAS Signaling

Journal: Current Medicinal Chemistry
Volume: 20 Issue: 31 Year: 2013 Page: 3944-3953
Author(s): Ting-Tsz Ou,Ming-Cheng Lin,Cheng-Hsun Wu,Wea-Lung Lin,Chau-Jong Wang

Anticancer Therapeutic Strategies Based on CDK Inhibitors

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 3 Year: 2013 Page: 5327-5332
Author(s): Luca Esposito, Paola Indovina, Flora Magnotti, Daniele Conti, Antonio Giordano

Glycogen Synthase Kinase 3 as an Anticancer Drug Target: Novel Experimental Findings and Trends in the Design of Inhibitors

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 4 Year: 2013 Page: 665-679
Author(s): Dmitry I. Osolodkin, Vladimir A. Palyulin, Nikolay S. Zefirov

Curcumin Potentiates The Ability of Sunitinib to Eliminate the VHL-lacking Renal Cancer Cells 786-O: Rapid Inhibition of Rb Phosphorylation as a Preamble to Cyclin D1 Inhibition

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 13 Issue: 10 Year: 2013 Page: 1508-1513
Author(s): Priya Ranjan Debata,Sultana Begum,Anita Mata,Oksana Genzer,Morton J. Kleiner,Probal Banerjee,Mario R. Castellanos

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