Search Result "conjugate addition"


Recent Advances in Site Specific Conjugations of Antibody Drug Conjugates (ADCs)

Journal: Current Cancer Drug Targets
Volume: 16 Issue: 6 Year: 2016 Page: 469-479
Author(s): Wenlong Gao,Jingxin Zhang,Jun Xiang,Lei Zhang,Chengbin Wu,Pradeep K. Dhal,Bo Chen

Nucleophilic Addition of Cyclopropenes

Journal: Current Organic Chemistry
Volume: 20 Issue: 1 Year: 2016 Page: 1862-1877
Author(s): Andrew Edwards, Marina Rubina, Michael Rubin

Polymer Drug Conjugates: Recent Advancements in Various Diseases

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 19 Year: 2016 Page: 2821-2843
Author(s): Jasbir Singh,Sapna Desai,Snehlata Yadav,Balasubramanian Narasimhan,Harmeet Kaur

Research Article

Synthesis and Biological Evaluations of Cytotoxic and Antiangiogenic Triterpenoids-Jacaranone Conjugates

Journal: Medicinal Chemistry
Volume: 12 Issue: 8 Year: 2016 Page: 775-785
Author(s): Hua Sun, Partick Y.K. Yue, Shao-Rong Wang, Lihong Huo, Ying Zhao, Songbo Xie, Jens V. Kringelum, Ole Lund, Olivier Taboureau, Jun Zhou, Ricky N. S. Wong, Wei-Shuo Fang

Chemosensitization of Prostate Carcinoma Cells with a Receptor-directed Smac Conjugate

Journal: Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2016 Page: 412-418
Author(s): Alexander Sturzu,Sumbla Sheikh,Hartmut Echner,Martin Deeg,Thomas Nägele,Christopher Weidenmaier,Christian Schwentner,Marius Horger,Ulrike Ernemann,Stefan Heckl

Formation of A Novel Purine Metabolite through CYP3A4 Bioactivation and Glutathione Conjugation

Journal: Drug Metabolism Letters
Volume: 10 Issue: 2 Year: 2016 Page: 144-150
Author(s): Julius L. Apuy, Cathie Xiang, Sarah Franc, Sayee G. Hegde, Robert Hubbard, Jingjing Zhao, Mehran F. Moghaddam

Design and Synthesis of New Conjugates of Bile Acids with Salicylic, Acetylsalicylic and Nicotinic Acids

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 4 Year: 2016 Page: 302-309
Author(s): Tomasz Pospieszny,Bogumił Brycki

Research Article

Bispecific Antibodies for Targeted Delivery of Dendritic Polyglycerol (dPG) Prodrug Conjugates

Journal: Current Cancer Drug Targets
Volume: 16 Issue: 7 Year: 2016 Page: 639-649
Author(s):

Design, Synthesis and Antiproliferative Activity of Novel Benzothiazole Derivatives Conjugated with Semicarbazone Scaffold

Journal: Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2016 Page: 489-498
Author(s): Guanglong Bao,Baoquan Du,Yuxiu Ma,Meng Zhao,Ping Gong,Xin Zhai

Prospects of Bacteriotherapy with Nanotechnology in Nanoparticledrug Conjugation Approach for Cancer Therapy

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 14 Year: 2016 Page: 1477-1494
Author(s): Ritu Raj,Surajit Das

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