Search Result "chloroquine"


Reversed Chloroquine Molecules as a Strategy to Overcome Resistance in Malaria

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2012 Page: 400-407
Author(s): David H. Peyton

Synthesis and In Vivo Antimalarial Activity of Quinoline/Mercaptopurine Conjugates

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 4 Year: 2012 Page: 361-366
Author(s): Nicolli Bellotti de Souza, Rafael Carvalhaes, Arturene Maria Lino do Carmo, Marcio Jose Martins Alves,Elaine Soares Coimbra, Sonia Maria Neumann Cupolilo, Clarice Abramo, Adilson David Da Silva

Molecular Modeling Studies, Synthesis and Biological Evaluation of Novel Plasmodium falciparum Lactate Dehydrogenase (pfLDH) Inhibitors

Journal: Anti-Infective Agents
Volume: 10 Issue: 1 Year: 2012 Page: 55-71
Author(s): Premlata K. Ambre, Raghuvir R. S. Pissurlenkar, Ashish S. Jagyasi, Ritesh A. Fule, Vijay Khedkar, Chandrashekar R. Barhate, Livia Vivas, Abhai K. Tripathi, David Sullivan, Richard Birkinshaw, R. Leo Brady, Krishna Iyer, Evans C. Coutinho

QSAR Studies of Some Substituted 1,3-Diaryl Propenone Derivatives as Plasmodium falciparum Growth Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 2 Year: 2012 Page: 153-162
Author(s): Nitendra K. Sahu, Sanjaykumar B. Bari, D. V. Kohli

Design, Synthesis and Anti-itch Activity Evaluation of Aromatic Amino Acid Derivatives as Gastrin-Releasing Peptide Receptor Antagonists

Journal: Medicinal Chemistry
Volume: 8 Issue: 5 Year: 2012 Page: 865-873
Author(s): Ri-Sheng Yao,Ting-Ting Li,Jun Xu,Lai-En Jiang,Ban-Feng Ruan

Design, Synthesis and In Vitro Antimalarial Evaluation of New Quinolinylhydrazone Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 2 Year: 2012 Page: 163-168
Author(s): Le Thi Thuy, Hoang Xuan Tien, Vu Dinh Hoang, Tran Khac Vu

Synthesis and Preliminary Evaluation of n.c.a. Iodoquine: A Novel Radiotracer with High Uptake in Cells with High ALDH1 Expression

Journal: Current Radiopharmaceuticals
Volume: 5 Issue: 1 Year: 2012 Page: 47-58
Author(s): Bennett B. Chin, Anita Hjelemand, Jeremy Rich, Haijing Song, Christopher Lascola, Robert Storms, Roger McLendon, Robert Reiman, Kim L. Greer, Scott D. Metzler, Darryl McDougald, Diana Dai, Ganesan Vaidyanathan

Cytotoxic Activity of Polysubstituted 7-chloro-4-quinolinylhydrazone Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 3 Year: 2012 Page: 251-256
Author(s): Raquel Carvalho Montenegro, Leticia Veras Lotufo, Manoel Odorico de Moraes, Claudia do O Pessoa, Felipe Augusto Rocha Rodrigues, Marcelle de Lima Ferreira Bispo, Bruna Abreu Freire, Carlos Roland Kaiser, Marcus Vinicius Nora de Souza

Structural Insight for Imidazopyridazines as Malarial Kinase PfPK7 Inhibitors Using QSAR Techniques

Journal: Medicinal Chemistry
Volume: 8 Issue: 4 Year: 2012 Page: 636-648
Author(s): Nitendra K. Sahu,D. V. Kohli

In Vitro Antimycobacterial Activity of New 7-Chloroquinoline Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 9 Issue: 2 Year: 2012 Page: 126-134
Author(s): Juan Bueno, Fernando A. Rojas Ruiz, Santiago Villabona Estupinan, Vladimir V. Kouznetsov

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