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HCN Channels Modulators: The Need for Selectivity

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 16 Year: 2016 Page: 1764-1791
Author(s): Maria Novella Romanelli,Laura Sartiani,Alessio Masi,Guido Mannaioni,Dina Manetti,Alessandro Mugelli,Elisabetta Cerbai

Implications of Dynamic Occupancy, Binding Kinetics, and Channel Gating Kinetics for hERG Blocker Safety Assessment and Mitigation

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 16 Year: 2016 Page: 1792-1818
Author(s): Robert A. Pearlstein,K. Andrew MacCannell,Gül Erdemli,Sarita Yeola,Gabriel Helmlinger,Qi-Ying Hu,Ramy Farid,William Egan,Steven Whitebread,Clayton Springer,Jeremy Beck,Hao-Ran Wang,Mateusz Maciejewski,Laszlo Urban,José S. Duca

Calcium Channel Blockade and Peroxisome Proliferator Activated Receptor γ Agonism Diminish Cognitive Loss and Preserve Endothelial Function During Diabetes Mellitus

Journal: Current Neurovascular Research
Volume: 13 Issue: 1 Year: 2016 Page: 33-44
Author(s): Swati Jain,B. M Sharma,Bhupesh Sharma

Research Article

Sodium Channel Blocking Activity and In-vivo Testing of New Phenylimidazole Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 9 Year: 2016 Page: 962-967
Author(s): Mirko Rivara, Manoj K. Patel, Alberto Rapalli, Valentina Zuliani

Research Article

Chalcone Derivatives Activate and Desensitize the Transient Receptor Potential Ankyrin 1 Cation Channel, Subfamily A, Member 1 TRPA1 Ion Channel: Structure-Activity Relationships in vitro and Anti-Nociceptive and Anti-inflammatory Activity in vivo

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 15 Issue: 8 Year: 2016 Page: 987-994
Author(s): Aniello Schiano Moriello, Livio Luongo, Francesca Guida, Michael S. Christodoulou, Dario Perdicchia, Sabatino Maione, Daniele Passarella, Vincenzo Di Marzo, Luciano De Petrocellis

Drug-induced Inhibition and Trafficking Disruption of ion Channels: Pathogenesis of QT Abnormalities and Drug-induced Fatal Arrhythmias

Journal: Current Cardiology Reviews
Volume: 12 Issue: 2 Year: 2016 Page: 141-154
Author(s): Luigi X. Cubeddu

Selected PET Radioligands for Ion Channel Linked Neuroreceptor Imaging: Focus on GABA, NMDA and nACh Receptors

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 16 Year: 2016 Page: 1830-1842
Author(s): Alina Kassenbrock,Neil Vasdev,Steven H. Liang

Research Article

Cnidarian Neurotoxic Peptides Affecting Central Nervous System Targets

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 16 Issue: 3 Year: 2016 Page: 173-182
Author(s):

Review Article

Multiple Non-Equivalent Interfaces Mediate Direct Activation of GABAA Receptors by Propofol

Journal: Current Neuropharmacology
Volume: 14 Issue: 7 Year: 2016 Page: 772-780
Author(s): Megan M. Eaton,Allison L. Germann,Ruby Arora,Lily Q. Cao,Xiaoyi Gao,Daniel J. Shin,Albert Wu,David C. Chiara,Jonathan B. Cohen,Joe Henry Steinbach,Alex S. Evers,Gustav Akk

Research Article

Glycyrrhizic Acid Ameliorates Cognitive Impairment in a Rat Model of Vascular Dementia Associated with Oxidative Damage and Inhibition of Voltage-Gated Sodium Channels

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 15 Issue: 8 Year: 2016 Page: 1001-1008
Author(s): Jie Guo, Chunxiao Yang, Jiajia Yang, Yang Yao

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