Search Result "antichagasic candidate"


Synthesis Optimization of Hydroxymethylnitrofurazone, an Antichagasic Candidate, Using 32 Factorial Design

Journal: Letters in Organic Chemistry
Volume: 7 Issue: 3 Year: 2010 Page: 191-195
Author(s): Gustavo H.G. Trossini, Jeanine Giarolla, Leandro de Rezende, Antonia T. do Amaral, Marcio H. Zaim, Roy E. Bruns, Elizabeth I. Ferreira

Molecular Modeling and Docking Application to Evaluate Cruzain Inhibitory Activity by Chalcones and Hydrazides

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 3 Year: 2014 Page: 249-255
Author(s): Drielli Gomes Vital,Marco Arribas,Gustavo Henrique Goulart Trossini

Anti-T. cruzi Agents: Our Experience in the Evaluation of More than Five Hundred Compounds

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 8 Issue: 1 Year: 2008 Page: 1355-1383
Author(s): Hugo Cerecetto, Mercedes Gonzalez

An Insight on Targets and Patented Drugs for Chemotherapy of Chagas Disease

Journal: Recent Patents on Anti-Infective Drug Discovery
Volume: 2 Issue: 1 Year: 2007 Page: 19-51
Author(s): Vilma G. Duschak, Alicia S. Couto

Review Article

An Overview of Recent Advances in Biological and Pharmaceutical Developments of Fluoro-containing Drugs

Journal: Current Organic Chemistry
Volume: 23 Issue: 26 Year: 2019 Page: 2916-2944
Author(s): Nader G. Khaligh,Hanna Abbo,Salam J.J. Titinchi,Mohd R. Johan

Natural and Synthetic Naphthoquinones Active Against Trypanosoma Cruzi: An Initial Step Towards New Drugs for Chagas Disease

Journal: Current Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2011 Page: 144-161
Author(s): Cristian O. Salas, Mario Faundez, Antonio Morello, Juan Diego Maya, Ricardo A. Tapia

Review Article

The Role of Nitro (NO2-), Chloro (Cl), and Fluoro (F) Substitution in the Design of Antileishmanial and Antichagasic Compounds

Journal: Current Drug Targets
Volume: 22 Issue: 4 Year: 2021 Page: 367-386
Author(s): Boniface Pone Kamdem,Ferreira Igne Elizabeth

Key Proteins in the Polyamine-Trypanothione Pathway as Drug Targets Against Trypanosoma cruzi

Journal: Current Medicinal Chemistry
Volume: 21 Issue: 15 Year: 2014 Page: 1757-1771
Author(s): J.D. Maya,C.O. Salas,B. Aguilera-Venegas,M.V. Diaz,R. Lopez-Munoz

High-throughput Drug Repositioning for the Discovery of New Treatments for Chagas Disease

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 15 Issue: 3 Year: 2015 Page: 182-193
Author(s): Carolina L. Bellera,Maria L. Sbaraglini,Dario E. Balcazar,Laura Fraccaroli,M. Cristina Vanrell,A. Florencia Casassa,Carlos A. Labriola,Patricia S. Romano,Carolina Carrillo,Alan Talevi

Pharmacokinetics of Hydroxymethylnitrofurazone and Its Parent Drug Nitrofurazone in Rabbits

Journal: Drug Metabolism Letters
Volume: 7 Issue: 1 Year: 2013 Page: 58-64
Author(s): Marco Antonio Ferraz Nogueira Filho,Elias Carvalho Padilha,Michel Leandro de Campos,Diego Vinicius de Pontes Machado,Marcelo Gomes Davanço,Kelly Christina Pestana,Chung Man Chin,Rosângela Gonçalves Peccinini

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