Search Result "amino-thiazole inhibitors"


Macrocyclic Histone Deacetylase Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1423-1440
Author(s): Sandra C. Mwakwari, Vishal Patil, William Guerrant, Adegboyega K. Oyelere

Development of Nitrile-Based Peptidic Inhibitors of Cysteine Cathepsins

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 3 Year: 2010 Page: 294-322
Author(s): Maxim Frizler, Marit Stirnberg, Mihiret Tekeste Sisay, Michael Gutschow

CDK Inhibitors: From the Bench to Clinical Trials

Journal: Current Drug Targets
Volume: 11 Issue: 3 Year: 2010 Page: 279-290
Author(s): Flavio Rizzolio, Tiziano Tuccinardi, Isabella Caligiuri, Chiara Lucchetti, Antonio Giordano

Structure Based Design of 11β-HSD1 Inhibitors

Journal: Current Pharmaceutical Biotechnology
Volume: 11 Issue: 7 Year: 2010 Page: 779-791
Author(s): Suresh B. Singh, Colin M. Tice

Recent Progress of Src SH2 and SH3 Inhibitors as Anticancer Agents

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2010 Page: 1117-1124
Author(s): X.-L. Lu, X. Cao, X.-Y. Liu, B.-H. Jiao

Tyrosine Kinase Inhibitors

Journal: Current Cancer Drug Targets
Volume: 10 Issue: 5 Year: 2010 Page: 462-483
Author(s): C. Natoli, B. Perrucci, F. Perrotti, L. Falchi, S. Iacobelli

Inhibitors of the Sphingosine Kinase Pathway as Potential Therapeutics

Journal: Current Cancer Drug Targets
Volume: 10 Issue: 4 Year: 2010 Page: 354-367
Author(s): M.R. Pitman, S.M. Pitson

Proteases of Plasmodium falciparum as Potential Drug Targets and Inhibitors Thereof

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 3 Year: 2010 Page: 346-367
Author(s): Christof Wegscheid-Gerlach, Hans-Dieter Gerber, Wibke E. Diederich

Recent Advances in Stearoyl-CoA Desaturase 1 Inhibitors for Dyslipidemia and Obesity

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 4 Year: 2010 Page: 419-433
Author(s): Gang Liu

The Recent Medicinal Chemistry Development of Jak2 Tyrosine Kinase Small Molecule Inhibitors

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2010 Page: 4551-4558
Author(s): R. Baskin, A. Majumder, P. P. Sayeski

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