Search Result "allosteric modulators"


Positive Allosteric Modulators for mGluR2 Receptors: A Medicinal Chemistry Perspective

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 15 Year: 2014 Page: 1771-1788
Author(s): Gyorgy Szabo,Gyorgy Miklos Keseru

SAR Studies on Carboxylic Acid Series M1 Selective Positive Allosteric Modulators (PAMs)

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 15 Year: 2014 Page: 1738-1754
Author(s): Scott D. Kuduk,Douglas C. Beshore

SAR Studies on mGlu5 Receptor Positive Allosteric Modulators (2003- 2013)

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 15 Year: 2014 Page: 1789-1841
Author(s): Junliang Hao,Hui Xiong

Editorial free to download

Editorial (Thematic Issue: Allosteric Modulators of G Protein-Coupled Receptors)

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 15 Year: 2014 Page: 1735-1737
Author(s): Gregory J. Wells

Druggable Orthosteric and Allosteric Hot Spots to Target Protein-protein Interactions

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 8 Year: 2014 Page: 1293-1301
Author(s): Buyong Ma, Ruth Nussinov

Positive Allosteric Modulators (PAMs) of Metabotropic Glutamate Receptor 5 (mGluR5) Attenuate Microglial Activation

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 13 Issue: 4 Year: 2014 Page: 558-566
Author(s): Fengtian Xue,Bogdan A. Stoica,Marie Hanscom,Shruti V. Kabadi,Alan I. Faden

Allosteric Inhibition of G-Protein Coupled Receptor Oligomerization: Strategies and Challenges for Drug Development

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 15 Year: 2014 Page: 1842-1863
Author(s): Mattan Hurevich,Alaa Talhami,Deborah E. Shalev,Chaim Gilon

Chemical Biology of mGlu4 Receptor Activation: Dogmas, Challenges, Strategies and Opportunities

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 15 Year: 2014 Page: 1755-1770
Author(s): Xinyan Huang,Elena Dale,Robbin M. Brodbeck,Dario Doller

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 3 Year: 2014 Page: 304-312
Author(s): Gregor J. Macdonald, Craig W. Lindsley

A Common Molecular Motif Characterizes Extracellular Allosteric Enhancers of GPCR Aminergic Receptors and Suggests Enhancer Mechanism of Action

Journal: Current Medicinal Chemistry
Volume: 21 Issue: 32 Year: 2014 Page: 3673-3686
Author(s): Robert Root-Bernstein,Patrick F. Dillon

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