Search Result "admet"


Research Article

In-silico & In-vitro Identification of Structure-Activity Relationship Pattern of Serpentine & Gallic Acid Targeting PI3Kγ as Potential Anticancer Target

Journal: Current Cancer Drug Targets
Volume: 17 Issue: 8 Year: 2017 Page: 722-734
Author(s): Pooja Sharma,Aparna Shukla,Komal Kalani,Vijaya Dubey,Suaib Luqman,Santosh Kumar Srivastava,Feroz Khan

Research Article

3D-QSAR, Virtual Screening, Docking and Design of Dual PI3K/mTOR Inhibitors with Enhanced Antiproliferative Activity

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 4 Year: 2017 Page: 292-303
Author(s): Jelena Oluić,Katarina Nikolic,Jelica Vucicevic,Zarko Gagic,Slavica Filipic,Danica Agbaba

Review Article

Helix-Coil Transition Signatures B-Raf V600E Mutation and Virtual Screening for Inhibitors Directed Against Mutant B-Raf

Journal: Current Drug Metabolism
Volume: 18 Issue: 6 Year: 2017 Page: 527-534
Author(s): Srinivas Bandaru,Tharaparambil Gangadharan Sumithnath,Saphy Sharda,Sanskruti Lakhotia,Anudeep Sharma,Amrita Jain,Tajamul Hussain,Anuraj Nayarisseri,Sanjeev Kumar Singh

Research Article

In Silico Prioritization, Synthesis and In Vitro Evaluation of Tembamide Analogs for Anti-HIV Activity

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 1455-1464
Author(s): Shiv Gupta, Sanjay Kumar, Nisha Jariwala, Deepali Bhadane, Kamlesh Kumar Bhutani, Smita Kulkarni, Inder Pal Singh

Research Article

Molecular Modelling of Berberine Derivatives as Inhibitors of Human Smoothened Receptor and Hedgehog Signalling Pathway Using a Newly Developed Algorithm on Anti-Cancer Drugs

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 12 Issue: 4 Year: 2017 Page: 384-400
Author(s): Parham Jabbarzadeh Kaboli,Mohammad Bazrafkan,Patimah Ismail,King-Hwa Ling

Research Article

Design, Synthesis and Biological Evaluation of a Phenyl Butyric Acid Derivative, N-(4-chlorophenyl)-4-phenylbutanamide: A HDAC6 Inhibitor with Anti-proliferative Activity on Cervix Cancer and Leukemia Cells

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 10 Year: 2017 Page: 1441-1454
Author(s): Rodriguez-Fonseca Rolando Alberto,Sixto-Lopez Yudibeth,Fragoso-Vazquez M. Jonathan,Flores-Mejia Raul,Cabrera-Perez Laura Cristina,Vazquez-Moctezuma Ismael,Rosales-Hernandez Martha Cecilia,Bello Martiniano,Martinez-Archundia M,Trujillo-Ferrara Jose Guadalupe,Becerra-Martinez Elvia,Correa-Basurto Jose

Research Article

In Silico Design, Synthesis and Bioactivity of N-(2, 4-Dinitrophenyl)-3-oxo- 3-phenyl-N-(aryl) Phenyl Propanamide Derivatives as Breast Cancer Inhibitors

Journal: Current Computer-Aided Drug Design
Volume: 13 Issue: 2 Year: 2017 Page: 112-126
Author(s): Mucheli Ramana,Rama Lokhande,Shanta Bhar,Prasanna Ranade,Ankita Mehta,Gayatri Gadre

Review Article

Recent Advances of Computational Modeling for Predicting Drug Metabolism: A Perspective

Journal: Current Drug Metabolism
Volume: 18 Issue: 1 Year: 2017 Page: 1106-1122
Author(s): Supratik Kar,Jerzy Leszczynski

Review Article

Recent Updates on Computer-aided Drug Discovery: Time for a Paradigm Shift

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 3296-3307
Author(s): Talambedu Usha,Dhivya Shanmugarajan,Arvind Kumar Goyal,Chinaga Suresh Kumar,Sushil Kumar Middha

Research Article

Molecular Docking and Molecular Dynamics Simulation Based Approach to Explore the Dual Inhibitor Against HIV-1 Reverse Transcriptase and Integrase

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 8 Year: 2017 Page: 734-746
Author(s): Subhash Chander,Rajan Kumar Pandey,Ashok Penta,Bhanwar Singh Choudhary,Manish Sharma,Ruchi Malik,Vijay Kumar Prajapati,Sankaranarayanan Murugesan

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