Search Result "T315I mutation"


Review Article

The Polyhedric Abl Kinases and their Pharmacologic Inhibitors

Journal: Current Enzyme Inhibition
Volume: 13 Issue: 2 Year: 2017 Page: 129-138
Author(s): Elisa Lupino, Marco Piccinini

Review Article

Insight to Pharmacokinetics of TKIs: Optimizing Practical Guidelines for Individualized Therapy

Journal: Current Drug Metabolism
Volume: 18 Issue: 3 Year: 2017 Page: 199-206
Author(s): Ruiqing Wang,Chaoqin Zhong,Chen Zhang,Mingqiang Hua,Daoxin Ma

Review Article

Recurrent Fusion Genes in Leukemia: An Attractive Target for Diagnosis and Treatment

Journal: Current Genomics
Volume: 18 Issue: 5 Year: 2017 Page: 378-384
Author(s): Yuhui Wang,Nan Wu,Duo Liu,Yan Jin

Review Article

Expanding the Opportunities for Modulating Kinase Targets with Allosteric Approaches

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 59-70
Author(s): Henrik Mobitz,Wolfgang Jahnke,Sandra W. Cowan-Jacob

Cancer Chemotherapy: Recent Developments in Hematology Oncology

Ebook: Frontiers in Drug Design & Discovery

Volume: 8 Year: 2017
Author(s): Sapna Parmar,Rebecca Nelson,Erica Hochard
Doi: 10.2174/9781681083551117080003
Research Article

In Vitro Sensitivity Profiling of Neuroblastoma Cells Against A Comprehensive Small Molecule Kinase Inhibitor Library to Identify Agents for Future Therapeutic Studies

Journal: Current Cancer Drug Targets
Volume: 17 Issue: 6 Year: 2017 Page: 569-584
Author(s): Anjali Singh,Vanessa Meier-Stephenson,Aarthi Jayanthan,Aru Narendran

Review Article

Stem Cell Guardians – Old and New Perspectives in LSC Biology

Journal: Current Drug Targets
Volume: 18 Issue: 4 Year: 2017 Page: 405-413
Author(s): Gillian A. Horne,Lorna Jackson,Vignir Helgason,Tessa L. Holyoake

Review Article

Unleashing the Guardian: The Targetable BCR-ABL/HAUSP/PML/PTEN Network in Chronic Myeloid Leukemia

Journal: Current Drug Targets
Volume: 18 Issue: 4 Year: 2017 Page: 389-395
Author(s): Alessandro Morotti,Davide Torti,Giovanna Carra,Cristina Panuzzo,Sabrina Crivellaro,Riccardo Taulli,Carmen Fava,Angelo Guerrasio,Giuseppe Saglio

Review Article

Cellular and Molecular Networks in Chronic Myeloid Leukemia: The Leukemic Stem, Progenitor and Stromal Cell Interplay

Journal: Current Drug Targets
Volume: 18 Issue: 4 Year: 2017 Page: 377-388
Author(s): Danilo Perrotti,Giovannino Silvestri,Lorenzo Stramucci,Justine Yu,Rossana Trotta

Review Article

Leveraging Structural Diversity and Allosteric Regulatory Mechanisms of Protein Kinases in the Discovery of Small Molecule Inhibitors

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 4 Year: 2017 Page: 4838-4872
Author(s): Gennady M. Verkhivker

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