Search Result "Structure-activity relationship."


Isothiocyanate Synthetic Analogs: Biological Activities, Structure-Activity Relationships and Synthetic Strategies

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 14 Issue: 12 Year: 2014 Page: 963-977
Author(s): Andrea Milelli,Carmela Fimognari,Nicole Ticchi,Paolo Neviani,Anna Minarini,Vincenzo Tumiatti

Synthesis, Structure-Activity Relationships and Biological Activity of New Isatin Derivatives as Tyrosinase Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 14 Issue: 12 Year: 2014 Page: 1450-1462
Author(s): Nahit Gencer,Fatih Sonmez,Dudu Demir,Oktay Arslan,Mustafa Kucukislamoglu

Structure Activity Relationships of Novel Antiepileptic Drugs

Journal: Current Medicinal Chemistry
Volume: 21 Issue: 6 Year: 2014 Page: 722-754
Author(s): G.K. Mittapalli,E. Roberts

Synthesis, Structure-Activity Relationship (SAR) Studies on some 4-Aryl-4Hchromenes and Relationship between Lipophilicity and Antitumor Activity

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 1 Year: 2014 Page: 1167-1176
Author(s): Ahmed M. El-Agrody, Essam Shawky A. E. H. Khattab, Ahmed M. Fouda

Synthesis and Structure Activity Relationship Study of N-substituted 3,5-diarylidenepiperidin- 4-ones as Potential Antitumor Agents

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 14 Issue: 2 Year: 2014 Page: 319-330
Author(s): Hala Bakr El-Nassan

Synthesis, Characterization and Structure Activity Relationship Studies of Benzo[b]thiophene Derivatives as Promising Class of Antimicrobial Agents

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 3 Year: 2014 Page: 349-354
Author(s): H.B. Ghodasara,R.G. Vaghasiya,V.K. Gothaliya,V.H. Shah

Research Article

Quantitative Structure Activity Relationship and Design of Phenyl Alkyl Ketone Derivatives as Inhibitors of Phosphodiesterase 4

Journal: Current Enzyme Inhibition
Volume: 10 Issue: 1 Year: 2014 Page: 68-80
Author(s): Anand Gaurav,Vertika Gautam,Ranjit Singh

Structural Studies on N-(1-naphthyl)-3-amino-5-oxo-4-phenyl-1Hpyrazole- 1-carboxamide with Antibacterial Activity

Journal: Letters in Organic Chemistry
Volume: 11 Issue: 1 Year: 2014 Page: 40-48
Author(s): Agnieszka A. Kaczor, Tomasz Wrobel, Zbigniew Karczmarzyk, Waldemar Wysocki, Andrzej Fruzinski, Malgorzata Brodacka, Dariusz Matosiuk, Monika Pitucha

Quantitative Structure-Retention Relationships Studies of Selected Groups of Compounds Characterized by Different Pharmacological Activity Using Multiple Linear Regression Procedure

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 8 Year: 2014 Page: 1017-1039
Author(s): Jolanta Stasiak,Marcin Koba,Tomasz Baczek

Relationship of Azole Resistance with the Structural Alteration of the Target Sites: Novel Synthetic Compounds for Better Antifungal Activities

Journal: The Natural Products Journal
Volume: 4 Issue: 2 Year: 2014 Page: 131-139
Author(s): Parth Malik,Narender Chaudhry,Bheru S. Kitawat,Raman Kumar,Tapan K. Mukherjee

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