Search Result "SAR-activity"


Novel High Throughput Polymer Biocompatibility Screening Designed for SAR (Structure-Activity Relationship): Application for Evaluating Polymer Coatings for Cardiovascular Drug-Eluting Stents

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 12 Issue: 7 Year: 2009 Page: 664-676
Author(s): Ayala Hezi-Yamit, Carol Sullivan, Jennifer Wong, Laura David, Mingfei Chen, Peiwen Cheng, David Shumaker, Josiah Wilcox, Kishore Udipi

Extraction of Structure-Activity Relationship Information from High-Throughput Screening Data

Journal: Current Medicinal Chemistry
Volume: 16 Issue: 3 Year: 2009 Page: 4049-4057
Author(s): M. Wawer, J. Bajorath

Structure-Activity Relationship (SAR): Effort Towards Blocking NGlucuronidation of Indazoles (PF-03376056) By Human UGT1A Enzymes

Journal: Drug Metabolism Letters
Volume: 3 Issue: 1 Year: 2009 Page: 28-34
Author(s): Kelly Rose, Young-Sun Yang, Richard Sciotti, Hongliang Cai

Pentacyclic Triterpenoids and Their Saponins with Apoptosis-Inducing Activity

Journal: Current Topics in Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2009 Page: 1581-1596
Author(s): Shao-Rong Wang, Wei-Shuo Fang

Structure-Based Design of Benzimidazole Sugar Conjugates: Synthesis, SAR and In Vivo Anti-inflammatory and Analgesic Activities

Journal: Medicinal Chemistry
Volume: 5 Issue: 6 Year: 2009 Page: 558-569
Author(s): Ahmed O.H. El-Nezhawy, Samir T. Gaballah, Mohamed A.A. Radwan, Ayman R. Baiuomy, Omar M.E. Abdel-Salam

Fentanyl Analogs: Structure-Activity-Relationship Study

Journal: Current Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2009 Page: 2468-2474
Author(s): S. Vuckovic, M. Prostran, M. Ivanovic, Lj. Dosen-Micovic, Z. Todorovic, Z. Nesic, R. Stojanovic, N. Divac, Z. Mikovic

Phenanthroindolizidines and Phenanthroquinolizidines: Promising Alkaloids for Anti-Cancer Therapy

Journal: Current Bioactive Compounds
Volume: 5 Issue: 1 Year: 2009 Page: 2-19
Author(s): Sherry R. Chemler

Small Molecule Aurora Kinases Inhibitors

Journal: Current Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2009 Page: 1949-1963
Author(s): Laura Garuti, Marinella Roberti, Giovanni Bottegoni

Urea Derivatives as Anticancer Agents

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 9 Issue: 4 Year: 2009 Page: 471-480
Author(s): Huan-Qiu Li, Peng-Cheng Lv, Tao Yan, Hai-Liang Zhu

Sulfanyltriazole/tetrazoles: A Promising Class of HIV-1 NNRTIs

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 8 Year: 2009 Page: 1014-1023
Author(s): Peng Zhan, Zhenyu Li, Xinyong Liu, Erik De Clercq

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