Search Result "QSAR study"


Research Article

Peptide Drugs QSAR Study Based on Topomer CoMFA

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 10 Year: 2017 Page: 1114-1121
Author(s): Jianbo Tong,Lingxiao Li,Kangnan Li,Min Bai

Review Article

The Role of QSAR and Virtual Screening Studies in Type 2 Diabetes Drug Discovery

Journal: Medicinal Chemistry
Volume: 13 Issue: 8 Year: 2017 Page: 706-720
Author(s): Simone Q. Pantaleao,Drielli G.V. Fujii,Vinicius G. Maltarollo,Danielle da C. Silva,Gustavo H.G. Trossini,Karen C. Weber,Luis P.B. Scott,Kathia M. Honorio

Research Article

Combined Approach of QSAR and Docking Studies for the Design of Local Anaesthetic Agents

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 3 Year: 2017 Page: 272-276
Author(s): Chunyan Zhang,Zhi Li,Jiahai Ma,Jing Zhang,Longming Zhang,Tao Li,Shijian Zheng

Research Article

Docking and QSAR Studies of 1,4-Dihydropyridine Derivatives as Anti- Cancer Agent

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 12 Issue: 2 Year: 2017 Page: 174-185
Author(s): Shirin Mollazadeh, Jamal Shamsara, Maryam Iman, Farzin Hadizadeh

Research Article

3D-QSAR Studies of Novel Cytotoxic Bufadienolides via CoMFA and CoMSIA Approaches

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 3 Year: 2017 Page: 306-313
Author(s): Hui Lin,Shengrong Li,Shiyao Li,Kangjia Liu,Yushui Han,Jialiang Guo,Longxin Lin,Yiqun Chang,Gaokeng Xiao,Weimin Chen,Pinghua Sun

Research Article

QSAR and Molecular Docking Studies on a Series of Cinnamic Acid Analogues as Epidermal Growth Factor Receptor (EGFR) Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 83-95
Author(s): Basheerulla Shaik,Omar Deeb,Vijay K. Agrawal,Satya P. Gupta

Research Article

Docking and QSAR Studies of Aryl-valproic Acid Derivatives to Identify Antiproliferative Agents Targeting the HDAC8

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 7 Year: 2017 Page: 927-940
Author(s): Heidy Martínez-Pacheco,Guillermo Ramírez-Galicia,Midalia Vergara-Arias,Jurg Gertsch,Jonathan Manuel Fragoso-Vazquez,David Mendez-Luna,A. L. Abujamra,Cabrera-Perez Laura Cristina,Rosales-Hernandez Martha Cecilia,I Mendoza-Lujambio,Jose Correa-Basurto

Research Article

Computational Screening of CCR5 Inhibitors as Potential Entry Inhibitor Microbicides Using 3D-QSAR Studies, Docking and Molecular Dynamics Simulation

Journal: Current HIV Research
Volume: 15 Issue: 4 Year: 2017 Page: 234-244
Author(s): Radhika Ramachandran,Muthusankar Aathi,Durairaj D. Ruban,Shanmughavel Piramanyagam

Research Article

Combined 3D-QSAR, Pharmacophore and Docking Studies on Benzenesulfonamide Derivatives as Potent 12-Lipoxygenase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 74-82
Author(s): Chunhong An,Mao Shu,Xiaoli Zai,Beina Zhang,Jing Li,Zichao Chang,Yong Hu,Zhihua Lin

Research Article

Docking-based 3D-QSAR Studies of Phosphodiesterase 9A Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 9 Year: 2017 Page: 986-998
Author(s): Changji Tan,Yinuo Wu,Yongxian Shao,Haibin Luo,Xuehua Zheng,Laiyou Wang

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