Search Result "QSAR"


Research Article

Novel 1,3,4-Triaryl Pyrazoles: Synthesis, QSAR Studies and Cytotoxicity against Breast Cancer

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 19 Issue: 7 Year: 2019 Page: 948-959
Author(s): Magda M. F. Ismail,Amel M. Farrag,Marwa F. Harras

Research Article

Novel Guanosine Derivatives as Anti-HCV NS5b Polymerase: A QSAR and Molecular Docking Study

Journal: Medicinal Chemistry
Volume: 15 Issue: 2 Year: 2019 Page: 130-137
Author(s): Abdo A. Elfiky

Research Article

DNA Cleavage Properties, Antimicrobial and Cytotoxic Activity and 4D-QSAR Analysis of Some Pyrazole Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 8 Year: 2019 Page: 904-918
Author(s): Semiha Kopru,Fatma Ozturk Küp,Nazmiye Sabanci,Mehmet Çadir,Duygu Cemre Bulut,Fatih Duman,Ilhan Ozer İlhan,Emin Saripinar

Research Article

DFT-Based QSAR Modelling of Inhibitory Activity of Coumarins and Sulfocoumarins on Carbonic Anhydrase (CA) Isoforms (CA I and CA II)

Journal: Current Computer-Aided Drug Design
Volume: 15 Issue: 3 Year: 2019 Page: 243-251
Author(s): Erol Eroglu

Research Article

3D QSAR Based Virtual Screening of Pyrido[1,2-a] Benzimidazoles as Potent Antimalarial Agents

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 3 Year: 2019 Page: 301-312
Author(s): Kalicharan Sharma,Apeksha Srivastava,Pooja Tiwari,Shweta Sharma,Mohammad Shaquiquzzaman,M. Mumtaz Alam,Mymoona Akhter

Research Article

Synthesis, Characterization, Antibacterial and Antioxidant Potency of NSubstituted- 2-Sulfanylidene-1,3-Thiazolidin-4-one Derivatives and QSAR Study

Journal: Medicinal Chemistry
Volume: 15 Issue: 8 Year: 2019 Page: 840-849
Author(s): Harshad Brahmbhatt,Maja Molnar,Valentina Pavić,Vesna Rastija

Research Article

QSAR Studies on Thiazole Derivatives as HCV NS5A Inhibitors via CoMFA and CoMSIA Methods

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 4 Year: 2019 Page: 453-460
Author(s): Jiayu Li,Wenyue Tian,Diaohui Gao,Yuying Li,Yiqun Chang,Jun Xu,Junxia Zheng,Pinghua Sun

Research Article

QSAR Analysis of Multimodal Antidepressants Vortioxetine Analogs Using Physicochemical Descriptors and MLR Modeling

Journal: Current Computer-Aided Drug Design
Volume: 15 Issue: 4 Year: 2019 Page: 294-307
Author(s): David M. Rajathei,Subbiah Parthasarathy,Samuel Selvaraj

Research Article

Discovery of New Phosphoinositide 3-kinase Delta (PI3Kδ) Inhibitors via Virtual Screening using Crystallography-derived Pharmacophore Modelling and QSAR Analysis

Journal: Medicinal Chemistry
Volume: 15 Issue: 6 Year: 2019 Page: 586-599
Author(s): Mahmoud A. Al-Sha`er,Rua`a A. Al-Aqtash,Mutasem O. Taha

Research Article

Synthesis, 2D-QSAR Studies and Biological Evaluation of Quinazoline Derivatives as Potent Anti-Trypanosoma cruzi Agents

Journal: Medicinal Chemistry
Volume: 15 Issue: 3 Year: 2019 Page: 265-276
Author(s): Mariela Bollini,Ana María Bruno,María Eugenia Niño,Juan José Casal,Leandro Daniel Sasiambarrena,Damián Ariel González Valdez,Leandro Battini,Vanesa Rocío Puente,María Elisa Lombardo

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