Search Result "QSAR"


Research Article

QSAR and Pharmacophore Mapping Studies on Benzothiazinimines to Relate their Structural Features with anti-HIV Activity

Journal: Medicinal Chemistry
Volume: 14 Issue: 7 Year: 2018 Page: 733-740
Author(s): Gopiraja Geethaavacini,Go Poh Poh,Lim Yi Yan,Rajindran Deepashini,Sivadasan Shalini,Rajak Harish,Krishnan Sureshkumar,Veerasamy Ravichandran

Review Article

Role of Topological, Electronic, Geometrical, Constitutional and Quantum Chemical Based Descriptors in QSAR: mPGES-1 as a Case Study

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2018 Page: 1075-1090
Author(s): Ashish Gupta,Virender Kumar,Polamarasetty Aparoy

Research Article

3D-QSAR Modeling of Some S-trityl-L-Cysteine Analogues as Inhibitors of Mitotic Kinesin Eg5 by CoMFA, CoMSIA and H-QSAR Methodologies

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 9 Year: 2018 Page: 979-987
Author(s): Fatemeh Mousavi,Mohammad Hossein Fatemi

Research Article

QSAR Analysis for Antioxidant Activity of Dipicolinic Acid Derivatives

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 21 Issue: 3 Year: 2018 Page: 204-214
Author(s): Vesna Rastija,Maja Molnar,Tena Siladi,Vijay Hariram Masand

Review Article

QSAR Modeling of Histamine H3R Antagonists/inverse Agonists as Future Drugs for Neurodegenerative Diseases

Journal: Current Neuropharmacology
Volume: 16 Issue: 6 Year: 2018 Page: 749-757
Author(s): Michelle Fidelis Correa,Joao Paulo dos Santos Fernandes

Research Article

Docking and 3D QSAR Studies on Substituted Cyclobutylphenyl Quinoline Derivatives as Inhibitors of Bacterial DNA Gyrase

Journal: Current Computer-Aided Drug Design
Volume: 14 Issue: 4 Year: 2018 Page: 322-337
Author(s): Rucha R. Wani,Hemchandra K. Chaudhari

Research Article

Atom-based and Pharmacophore-based 3D – QSAR Studies on Vitamin D Receptor (VDR)

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 21 Issue: 5 Year: 2018 Page: 329-343
Author(s): Selvaraman Nagamani,Chandrasekhar Kesavan,Karthikeyan Muthusamy

Research Article

2D & 3D-QSAR Study on Novel Piperidine and Piperazine Derivatives as Acetylcholinesterase Enzyme Inhibitors

Journal: Current Computer-Aided Drug Design
Volume: 14 Issue: 4 Year: 2018 Page: 391-397
Author(s): Maryam Nazari,Sayyed Abbas Tabatabai,Elham Rezaee

Research Article

The Quantum Chemical and QSAR Studies on Acinetobacter Baumannii Oxphos Inhibitors

Journal: Medicinal Chemistry
Volume: 14 Issue: 3 Year: 2018 Page: 253-268
Author(s): Hakan Sezgin Sayiner,Afaf A.S. Abdalrahm,Murat A. Basaran,Vasyl Kovalishyn,Fatma Kandemirli

Research Article

Pharmacophore and 3D-QSAR Characterization of Thieno[3,2-d] pyrimidine-6-carboxamides as SIRT-2 Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 6 Year: 2018 Page: 661-670
Author(s): Neetu Agrawal,Kamal Shah,Pradeep Mishra

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