Search Result "Pyrimidine derivatives"


Conjugates of 1,2,3-Triazoles and Acyclic Pyrimidine Nucleoside Analogues: Syntheses and X-ray Crystallographic Studies

Journal: Current Organic Chemistry
Volume: 17 Issue: 1 Year: 2013 Page: 1114-1124
Author(s): Silvija Korunda, Svjetlana Kristafor, Mario Cetina, Silvana Raic-Malic

Novel 2-hydrazino-pyrimidin-4(3H)-one Derivatives with Pseudofunctional- Similarity to Siderophores as Potential Antimycobacterial Agents

Journal: Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2013 Page: 77-83
Author(s): Ranjeet Bairwa, Nilesh R. Tawari, Amruta Alate, Swapnil Anam, Mariam S. Degani, Muktikant Ray, Ramakrishna M. G. Rajan

Synthesis and Antioxidant Activity of 1,2,4-Triazole linked Thieno[2,3- d]pyrimidine Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 10 Issue: 2 Year: 2013 Page: 186-193
Author(s): Suresh Maddila,Avula S. Kumar,Sridevi Gorle,M. Singh,Palakondu Lavanya,S.B. Jonnalagadda

6-Acetyl-5H-thiazolo[3,2-a]pyrimidine Derivatives as the Novel Acetylcholinesterase Inhibitors: Design, Synthesis, and Biological Activity

Journal: Medicinal Chemistry
Volume: 9 Issue: 5 Year: 2013 Page: 703-709
Author(s): Hui Zhi,Can Zhang,Zhixin Cheng,Zhe Jin,Erfang Huang,Shuo Li,Huangquan Lin,David Chicheong Wan,Chun Hu

Ionic Liquid Mediated Synthesis of Novel tetrahydroimidazo [1,2- a]pyrimidine-6-carboxylate Derivatives

Journal: Letters in Organic Chemistry
Volume: 10 Issue: 3 Year: 2013 Page: 178-184
Author(s): Vinod V. Thorat, Satish A. Dake, Satish U. Deshmukh, Elayaraja Rasokkiyam, Mohd. Farees Uddin, Rajendra P. Pawar

Thienyl Pyrimidine Derivatives with PrPSc Oligomer-Inducing Activity are a Promising Tool to Study Prions

Journal: Current Topics in Medicinal Chemistry
Volume: 13 Issue: 19 Year: 2013 Page: 2477-2483
Author(s): Thibaut Imberdis,Adeline Ayrolles-Torro,Jean-Michel Verdier,Véronique Perrier

Synthesis and Biological Evaluation of Some Novel Thieno[2,3-d] pyrimidine Derivatives as Potential Anti-inflammatory and Analgesic Agents

Journal: Medicinal Chemistry
Volume: 9 Issue: 8 Year: 2013 Page: 1099-1112
Author(s): Alaa A. El-Tombary,Soad A.M. El-Hawash,Nargues S. Habib,Raafat Soliman,Ibrahim M. El-Ashmawy,Omaima G. Shaaban

One-Pot Synthesis of 5-Unsubstituted-6-Aroyl[1,2,4]triazolo[1,5-a]pyrimidine Utilizing Biginelli-Like Multicomponent Reaction of Enaminones with 3-Amino-1,2,4- triazole as the Urea Component

Journal: Current Organic Synthesis
Volume: 10 Issue: 6 Year: 2013 Page: 974-976
Author(s): Huwaida M.E. Hassaneen,Ismail A. Abdelhamid

Synthesis of 3-(2-chloroethyl)-2-methyl-6,7,8,9-tetrahydro-4H-pyrido[1,2- a] pyrimidin-4-one Derivatives as Antibacterial Agents

Journal: Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2013 Page: 240-248
Author(s): Byregowda Krishnamurthy,Kambappa Vinaya,Devraj Rakshith,Doddakunche Shivaramu Prasanna,Kanchugarakoppal Subbegowda Rangappa

Antiepileptic Activity of Novel 2-(substituted benzylidene)-7-(4- fluorophenyl)-5-(furan-2-yl)-2H-thiazolo[3,2-a]pyrimidin-3(7H)-one Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 10 Issue: 3 Year: 2013 Page: 204-211
Author(s): T. Panneer Selvam,V. Karthick,P. Vijayaraj Kumar,M. Ashraf Ali

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