Search Result "Pyrimidine derivatives"


A Novel Biginelli-Like Reaction: An Efficient One-pot Synthesis of Spiro[oxindole-quinazoline/pyrimidine]ones

Journal: Letters in Organic Chemistry
Volume: 7 Issue: 4 Year: 2010 Page: 277-282
Author(s): Hassan Kefayati, Kurosh Rad-Moghadam, Masoumeh Zamani, Sanaz Hosseyni

Evaluation of Novel 7-(hetero)aryl-substituted Pyrazolo[1, 5-a]pyrimidines as Phosphodiesterase-4 Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 7 Issue: 6 Year: 2010 Page: 402-408
Author(s): Arumugam Kodimuthali, Rajesh Gupta, Kishore Venkata Laxmi Parsa, Padala Lakshmi Prasunamba, Manojit Pal

Inhibitors of the Mitochondrial Electron Transport Chain and de novo Pyrimidine Biosynthesis as Antimalarials: The Present Status

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2010 Page: 929-956
Author(s): T. Rodrigues, F. Lopes, R. Moreira

Synthesis of N-Glucopyranosidic Derivatives as Potential Inhibitors that Bind at the Catalytic Site of Glycogen Phosphorylase

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1127-1138
Author(s): T. Gimisis

Pyrimidine Nucleosides in Molecular PET Imaging of Tumor Proliferation

Journal: Current Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2010 Page: 1010-1029
Author(s): M. M. Alauddin, J. G. Gelovani

α-Hydroxyiminophosphonate, -phosphinate and -phosphonium Derivatives

Journal: Current Organic Synthesis
Volume: 7 Issue: 6 Year: 2010 Page: 628-649
Author(s): Javier Vicario, Concepcion Alonso, Jesus M. de los Santos, Francisco Palacios

Synthesis of Purine Derivatives as Scaffolds for a Diversity of Biological Activities

Journal: Current Organic Chemistry
Volume: 14 Issue: 2 Year: 2010 Page: 2463-2482
Author(s): A. Conejo-Garcia, O. Cruz-Lopez, V. Gomez-Perez, F. Morales, M. E. Garcia-Rubino, M. Kimatrai, M. C.Nunez, J. M. Campos

Cyclin-Dependent Kinase 4/6 (Cdk4/6) Inhibitors: Perspectives in Cancer Therapy and Imaging

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 10 Issue: 6 Year: 2010 Page: 527-539
Author(s): F. Graf, B. Mosch, L. Koehler, R. Bergmann, F. Wuest, J. Pietzsch

Recent Developments of Thalidomide Derivatives Possessing Anti-Inflammatory Activity

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2010 Page: 71-81
Author(s): Hulya Akgun, Irem Karamelekoglu

Development of Integrase Inhibitors of Quinolone Acid Derivatives for Treatment of AIDS: An Overview

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 10 Issue: 1 Year: 2010 Page: 1046-1057
Author(s): Z. G. Luo, J. J. Tan, Y. Zeng, C. X. Wang, L. M. Hu

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