Search Result "Protein kinase"


Exploiting Substrate Recognition for Selective Inhibition of Protein Kinases

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 20 Year: 2012 Page: 2914-2920
Author(s): Avital Licht-Murava,Hagit Eldar-Finkelman

Targeting Protein Kinases in the Malaria Parasite: Update of an Antimalarial Drug Target

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2012 Page: 456-472
Author(s): Veronica M. Zhang, Marina Chavchich, Norman C. Waters

New Insights in Protein Kinase Conformational Dynamics

Journal: Current Topics in Medicinal Chemistry
Volume: 12 Issue: 17 Year: 2012 Page: 1889-1895
Author(s): Giorgio Saladino,Francesco Luigi Gervasio

Conformationally Constrained Peptides as Protein Tyrosine Kinase Inhibitors

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 20 Year: 2012 Page: 2852-2866
Author(s): Rakesh K. Tiwari,Keykavous Parang

Recent Advances in Designing Substrate-Competitive Protein Kinase Inhibitors

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 20 Year: 2012 Page: 2875-2882
Author(s): Ki-Cheol Han,So Yeon Kim,Eun Gyeong Yang

New Directions in Targeting Protein Kinases: Focusing Upon True Allosteric and Bivalent Inhibitors

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 20 Year: 2012 Page: 2936-2945
Author(s): Vandana Lamba,Indraneel Ghosh

Synthesis of Cis-Fused Pyran Indolocarbazole Derivatives that Inhibit FLT3 Kinase and the DNA Damage Kinase, Checkpoint Kinase 1

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 12 Issue: 3 Year: 2012 Page: 194-201
Author(s): Francoise M. Perron-Sierra, Nathalie Kucharkzyk, Celine Boucley, Christel Guyard-Daumas, Sophie Sciberras, Christine Fouache, Sabine Plantier, Aurelie Studeny, Celine Bossard, Patrick J. Casara, Roy M. Golsteyn

Potential Role of Rho-Associated Protein Kinase Inhibitors for Glaucoma Treatment

Journal: Recent Patents on Endocrine, Metabolic & Immune Drug Discovery
Volume: 6 Issue: 2 Year: 2012 Page: 89-98
Author(s): Basilio Colligris,Almudena Crooke,Fernando Huete,Jesus Pintor

Novel Patented Src Kinase Inhibitor

Journal: Current Medicinal Chemistry
Volume: 19 Issue: 12 Year: 2012 Page: 1821-1829
Author(s): Xiao-Ling Lu,Xiao-Yu Liu,Xin Cao,Bing-Hua Jiao

Cis-enone Resorcylic Acid Lactones (RALs) as Irreversible Protein Kinase Inhibitors

Journal: Current Pharmaceutical Design
Volume: 18 Issue: 9 Year: 2012 Page: 1186-1198
Author(s): Linyi Wei, Jiuhong Wu, Guanqun Li, Ning Shi

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