Search Result "PI3K�� inhibitors"


Advances in the Development of Class I Phosphoinositide 3-Kinase (PI3K) Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 13 Year: 2016 Page: 1413-1426
Author(s): Dima A. Sabbah,Jian Hu,Haizhen A. Zhong

Review Article

Triggering PIK3CA Mutations in PI3K/Akt/mTOR Axis: Exploration of Newer Inhibitors and Rational Preventive Strategies

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 39 Year: 2016 Page: 6039-6054
Author(s): Vivek Asati,Sanjay K. Bharti,Debarshi Kar Mahapatra,Vikas Asati,Ashok K. Budhwani

Research Article

Review of PI3K/mTOR Inhibitors Entering Clinical Trials to Treat Triple Negative Breast Cancers

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 11 Issue: 3 Year: 2016 Page: 283-296
Author(s): Amélie Fouqué,Mickael Jean,Pierre van de Weghe,Patrick Legembre

Targeting the PI3K/AKT/mTOR Pathway in Prostate Cancer Development and Progression: Insight to Therapy

Journal: Clinical Cancer Drugs
Volume: 3 Issue: 1 Year: 2016 Page: 36-62
Author(s): Festuccia Claudio

Review Article

An Overview on Small Molecule Inhibitors of BRD4

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2016 Page: 1403-1414
Author(s): Wenhai Huang, Xiaoliang Zheng, Yewei Yang, Xiaoju Wang, Zhengrong Shen

Benzofuran Small Molecules as Potential Inhibitors of Human Protein Kinases. A Review

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 7 Year: 2016 Page: 879-894
Author(s): Halina Kwiecień,Agata Goszczyńska,Paulina Rokosz

Overcoming Resistance to EGFR Inhibitors in NSCLC

Journal: Reviews on Recent Clinical Trials
Volume: 11 Issue: 2 Year: 2016 Page: 99-105
Author(s): Paolo Maione, Paola C. Sacco, Francesca Casaluce, Assunta Sgambato, Giuseppe Santabarbara, Antonio Rossi, Cesare Gridelli

Getting a Handle on RAS-targeted Therapies: Cysteine Directed Inhibitors

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 5 Year: 2016 Page: 383-390
Author(s): Minh V. Huynh,Sharon L. Campbell

Old Tyrosine Kinase Inhibitors and Newcomers in Gastrointestinal Cancer Treatment

Journal: Current Cancer Drug Targets
Volume: 16 Issue: 2 Year: 2016 Page: 175-185
Author(s): Erika Giordani,Federica Zoratto,Martina Strudel,Anselmo Papa,Luigi Rossi,Marina Minozzi,Davide Caruso,Eleonora Zaccarelli,Monica Verrico,Silverio Tomao

Nitric Oxide Synthase (NOS) Inhibitors in Cancer Angiogenesis

Journal: Current Enzyme Inhibition
Volume: 12 Issue: 1 Year: 2016 Page: 49-66
Author(s): Amit K. Halder,Avinaba Mukherjee,Nilanjan Adhikari,Achintya Saha,Tarun Jha

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