Search Result "NPS antagonists"


Review Article

Natural Steroids and Androgen Antagonists used as Neuroprotection in Common Neurological Disorders

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 16 Issue: 7 Year: 2017 Page: 763-771
Author(s): David Calderon Guzman,Hugo Juarez Olguin,Ernestina Hernandez Garcia,Monica Punzo Soto,Mayra Santillan Garcia,Gerardo Barragan Mejia

The Controversial Role of Adenosine A2A Receptor Antagonists as Neuro-protective Agents

Journal: Current Medicinal Chemistry - Central Nervous System Agents
Volume: 4 Issue: 1 Year: 2004 Page: 35-45
Author(s): Patrizia Popoli, David Blum, Annita Pintor, Maria Teresa Tebano, Claudio Frank, Marco Gianfriddo, Maria Rosaria Domenici, Serge N. Schiffmann, Felicita Pedata

Homology Modeling of Adenosine A2A Receptor and Molecular Docking for Exploration of Appropriate Potent Antagonists for Treatment of Parkinsons Disease

Journal: Current Aging Science
Volume: 2 Issue: 2 Year: 2009 Page: 127-134
Author(s): Vijai Singh, Pallavi Somvanshi

Melanin-Concentrating Hormone Receptor 1 Antagonists: A New Perspective for the Pharmacologic Treatment of Obesity

Journal: Current Medicinal Chemistry
Volume: 15 Issue: 1 Year: 2008 Page: 1025-1043
Author(s): Gildardo Rivera, Virgilio Bocanegra-Garcia, Silvia Galiano, Nuria Cirauqui, Javier Ceras, Silvia Perez, Ignacio Aldana, Antonio Monge

A2A Adenosine Receptor and its Modulators: Overview on a Druggable GPCR and on Structure-Activity Relationship Analysis and Binding Requirements of Agonists and Antagonists

Journal: Current Pharmaceutical Design
Volume: 14 Issue: 1 Year: 2008 Page: 1525-1552
Author(s): G. Cristalli, C. Lambertucci, G. Marucci, R. Volpini, D. Dal Ben

Vitronectin Receptor -αVβ3 Integrin- Antagonists: Chemical and Structural Requirements for Activity and Selectivity

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 2 Issue: 6 Year: 2002 Page: 531-542
Author(s): Christophe Henry, Nicolas Moitessier, Yves Chapleur

Research Article

CXCR4-targeted Nanoparticles Reduce Cell Viability, Induce Apoptosis and Inhibit SDF-1α Induced BT-549-Luc Cell Migration In Vitro

Journal: Current Drug Delivery
Volume: 14 Issue: 8 Year: 2017 Page: 1060-1070
Author(s): Chuda Chittasupho,Prartana Kewsuwan,Takashi Murakami

Non Peptidic αvβ3 Antagonists: Recent Developments

Journal: Current Medicinal Chemistry
Volume: 12 Issue: 1 Year: 2005 Page: 51-70
Author(s): Barbara Cacciari, Giampiero Spalluto

Research Article

Synthesis of Arylpiperazine Derivatives as Protease Activated Receptor 1 Antagonists and Their Evaluation as Antiproliferative Agents

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 7 Year: 2017 Page: 973-981
Author(s): Andrea Ilaria Zotti,Elena Di Gennaro,Angela Corvino,Francesco Frecentese,Elisa Magli,Elisa Perissutti,Giuseppe Cirino,Fiorentina Roviezzo,Manuela Terranova-Barberio,Federica Iannelli,Giuseppe Caliendo,Vincenzo Santagada,Ferdinando Fiorino,Alfredo Budillon,Beatrice Severino

Medicinal Chemical and Pharmacological Aspects of Imidazole-Containing Histamine H3 Receptor Antagonists

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 4 Issue: 9 Year: 2004 Page: 965-977
Author(s): Holger Stark, Markus Kathmann, Eberhard Schlicker, Walter Schunack, Birgit Schlegel, Wolfgang Sippl

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