Search Result "MDR1"


Small Molecule Inhibitors of Multidrug Resistance Gene (MDR1) Expression: Preclinical Evaluation and Mechanisms of Action

Journal: Current Cancer Drug Targets
Volume: 13 Issue: 8 Year: 2013 Page: 814-828
Author(s): Sofia A. Santos,Alexandra Paulo

Pregnane X Receptor (PXR) at the Crossroads of Human Metabolism and Disease

Journal: Current Drug Metabolism
Volume: 14 Issue: 3 Year: 2013 Page: 341-350
Author(s): Ioannis Koutsounas,Stamatios Theocharis,Efstratios Patsouris,Constantinos Giaginis

An overview of ABC and SLC Drug Transporter Gene Regulation

Journal: Current Drug Metabolism
Volume: 14 Issue: 2 Year: 2013 Page: 253-264
Author(s): Qiu-Xia Chen,Hai-Hong Hu,Quan Zhou,Ai-Ming Yu,Su Zeng

P-glycoprotein Inhibition as a Therapeutic Approach for Overcoming Multidrug Resistance in Cancer: Current Status and Future Perspectives

Journal: Current Cancer Drug Targets
Volume: 13 Issue: 3 Year: 2013 Page: 326-346
Author(s): Ziyad Binkhathlan, Afsaneh Lavasanifar

Hurdles with Using In Vitro Models to Predict Human Blood-brain Barrier Drug Permeability: A Special Focus on Transporters and Metabolizing Enzymes

Journal: Current Drug Metabolism
Volume: 14 Issue: 1 Year: 2013 Page: 120-136
Author(s): Ramzi Shawahna,Xavier Decleves,Jean-Michel Scherrmann

Pharmacogenetics, Pharmacogenomics and Epigenetics of Nrf2-regulated Xenobioticmetabolizing Enzymes and Transporters by Dietary Phytochemical and Cancer Chemoprevention

Journal: Current Drug Metabolism
Volume: 14 Issue: 6 Year: 2013 Page: 688-694
Author(s): Tien-Yuan Wu, Tin Oo Khor, Jong Hun Lee, Ka Lung Cheung, Limin Shu, Chi Chen, Ah-Ng Kong

Mechanisms of Drug Resistance in Cancer Chemotherapy: Coordinated Role and Regulation of Efflux Transporters and Metabolizing Enzymes

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 4 Year: 2013 Page: 7126-7140
Author(s): Ramya Krishna Vadlapatla, Aswani Dutt Vadlapudi, Dhananjay Pal, Ashim K. Mitra

Conventional Chemotherapy and Emerging Targeted Therapy for Advanced Adrenocortical Carcinoma

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 13 Issue: 2 Year: 2013 Page: 248-253
Author(s): Yun-Ze Xu,Yu Zhu

New Insight into P-Glycoprotein as a Drug Target

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 13 Issue: 1 Year: 2013 Page: 159-170
Author(s): Albert Breier,Lenka Gibalova,Mario Seres,Miroslav Barancik,Zdenka Sulova

Potential Application of Network Descriptions for Understanding Conformational Changes and Protonation States of ABC Transporters

Journal: Current Pharmaceutical Design
Volume: 19 Issue: 2 Year: 2013 Page: 4155-4172
Author(s): Tamas Hegedus, Gergely Gyimesi, Merse E. Gaspar, Kristof Z. Szalay, Rajeev Gangal, Peter Csermely

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