Search Result "JAK3-specific inhibitor"


Research Article

Transforming Mutations of Jak3 (A573V and M511I) Show Differential Sensitivity to Selective Jak3 Inhibitors

Journal: Clinical Cancer Drugs
Volume: 3 Issue: 2 Year: 2016 Page: 131-137
Author(s): G. Steven Martinez, Jeremy A. Ross, Robert A. Kirken

Anaplastic Lymphoma Kinase Inhibitors in Non-Small Cell Lung Cancer

Journal: Current Drug Targets
Volume: 17 Issue: 6 Year: 2016 Page: 739-745
Author(s): David M. Straughan, Sa d C. Azoury, Vivek Shukla

Insights into the Structural Features Essential for JAK2 Inhibition and Selectivity

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 13 Year: 2016 Page: 1331-1355
Author(s): Chao Zhao,Daulat Bikram Khadka,Won-Jea Cho

Cinnamic Acid Derivatives as Inhibitors of Oncogenic Protein Kinases – Structure, Mechanisms and Biomedical Effects#

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 10 Year: 2016 Page: 954-982
Author(s): Marcin Mielecki,Bogdan Lesyng

Clinical Confirmation that the Selective JAK1 Inhibitor Filgotinib (GLPG0634) has a Low Liability for Drug-drug Interactions

Journal: Drug Metabolism Letters
Volume: 10 Issue: 1 Year: 2016 Page: 38-48
Author(s): Florence Namour,Julie Desrivot,Annegret Van der Aa,Pille Harrison,Gerben van`t Klooster,Chantal Tasset

Review Article

Pharmacological Activation of Protein Phosphatase 2 A (PP2A): A Novel Strategy to Fight Against Human Malignancies?

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 3 Year: 2016 Page: 4286-4296
Author(s):

Review Article

Interferon Therapy in Lung Cancer: Current Perspectives

Journal: Current Cancer Therapy Reviews
Volume: 12 Issue: 4 Year: 2016 Page: 237-245
Author(s): Debosree Ghosh, Pratap Parida

Identification of Inflammatory, Metabolic, and Cell Survival Pathways Contributing to Cerebral Small Vessel Disease by Postmortem Gene Expression Microarray

Journal: Current Neurovascular Research
Volume: 13 Issue: 1 Year: 2016 Page: 58-67
Author(s): Marie-Françoise Ritz,Caspar Grond-Ginsbach,Manja Kloss,Markus Tolnay,Felix Fluri,Leo H. Bonati,Christopher Traenka,Thomas Zeis,Nicole Schaeren-Wiemers,Nils Peters,Stefan Thomas Engelter,Philippe Alexandre Lyrer

Review Article

Immunoregulatory and Effector Activities of Nitric Oxide and Reactive Nitrogen Species in Cancer

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 2 Year: 2016 Page: 2618-2636
Author(s): Cinzia Fionda, Maria Pia Abruzzese, Angela Santoni, Marco Cippitelli

Computer Aided Drug Design: Success and Limitations

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 5 Year: 2016 Page: 572-581
Author(s):

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