Search Result "JAK3-specific inhibitor"


Targeting JAK3 Tyrosine Kinase-Linked Signal Transduction Pathways with Rationally-Designed Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 7 Issue: 6 Year: 2007 Page: 612-623
Author(s): Fatih M. Uckun, Alexei Vassilev, Ilker Dibirdik, Heather Tibbles

Design of a Peptide Inhibitor of Tyrosine Kinase 2

Journal: Protein & Peptide Letters
Volume: 21 Issue: 5 Year: 2014 Page: 419-425
Author(s): Melissa G. Works,Benben Song,Patrick Kibler,Mary J. Tanga,Amit K. Galande,Annalisa D’Andrea

Review Article

Irreversible Kinase Inhibitors Targeting Cysteine Residues and their Applications in Cancer Therapy

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 1732-1753
Author(s): Debasis Das,Jian Hong

Therapeutic Potential of Janus Kinase 3 (JAK3) Inhibitors

Journal: Current Pharmaceutical Design
Volume: 10 Issue: 1 Year: 2004 Page: 1767-1784
Author(s): M. Cetkovic-Cvrlje, H. E. Tibbles

Tyrosine Kinase Inhibitors for the Treatment of Rheumatoid Arthritis

Journal: Current Topics in Medicinal Chemistry
Volume: 13 Issue: 6 Year: 2013 Page: 760-773
Author(s): Jose A. Gomez-Puerta, Attila Mocsai

Discovery of Notch-Sparing γ-Secretase Inhibitors

Journal: Current Alzheimer Research
Volume: 7 Issue: 3 Year: 2010 Page: 207-209
Author(s): C.E. Augelli-Szafran, H.-X. Wei, D. Lu, J. Zhang, Y. Gu, T. Yang, P. Osenkowski, W. Ye, M.S. Wolfe

Review Article

Novel Therapeutic Approaches in Rheumatoid Arthritis: Role of Janus Kinases Inhibitors

Journal: Current Medicinal Chemistry
Volume: 26 Issue: 1 Year: 2019 Page: 2823-2843
Author(s): Felice Rivellese,Antonio Lobasso,Letizia Barbieri,Bianca Liccardo,Amato de Paulis,Francesca Wanda Rossi

Review Article

Aurora Kinase Inhibitors in Head and Neck Cancer

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 3 Year: 2018 Page: 199-213
Author(s): Guangying Qi,Jing Liu,Sisi Mi,Takaaki Tsunematsu,Shengjian Jin,Wenhua Shao,Tian Liu,Naozumi Ishimaru,Bo Tang,Yasusei Kudo

JAK2 Inhibitors for Myelofibrosis: Why are They Effective in Patients with and Without JAK2V617F Mutation?

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 12 Issue: 9 Year: 2012 Page: 1098-1109
Author(s): Fabio P. S. Santos,Srdan Verstovsek

The 2010 Patent Landscape for Spleen Tyrosine Kinase Inhibitors+

Journal: Recent Patents on Inflammation & Allergy Drug Discovery
Volume: 6 Issue: 2 Year: 2012 Page: 97-120
Author(s): Alessandro F. Moretto,Christoph Dehnhardt,Neelu Kaila,Nikolaos Papaioannou,Atli Thorarensen

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