Search Result "Inverse agonism"


A Pharmacological Primer of Biased Agonism

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 92-98
Author(s): Bradley T. Andresen

Histamine H3 Receptor (H3R) Antagonists and Inverse Agonists in the Treatment of Sleep Disorders

Journal: Current Pharmaceutical Design
Volume: 17 Issue: 1 Year: 2011 Page: 1426-1429
Author(s): Meredith Broderick, Tony Masri

The Evolution of Histamine H3 Antagonists/Inverse Agonists

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 6 Year: 2011 Page: 648-660
Author(s): Evan P. Lebois, Carrie K. Jones, Craig W. Lindsley

β-arrestin-Biased Agonism at the Parathyroid Hormone Receptor Uncouples Bone Formation from Bone Resorption

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 112-119
Author(s): Brittany N. Bohinc, Diane Gesty-Palmer

GABAA Receptor Subtype-Selective Modulators. II. α5-Selective Inverse Agonists for Cognition Enhancement

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 9 Year: 2011 Page: 1203-1214
Author(s): John R. Atack

Effects of Imidazolic Agonism on Blood Pressure, Sympathetic Activity, Left Ventricular Hypertrophy and Insulin Resistance

Journal: Current Hypertension Reviews
Volume: 7 Issue: 2 Year: 2011 Page: 88-94
Author(s): J. Soler, Maria J. Sanchez, R. A. Sanchez, A. J. Ramirez

Endogenous Ligand Bias by Chemokines: Implications at the Front Lines of Infection and Leukocyte Trafficking

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 11 Issue: 2 Year: 2011 Page: 120-131
Author(s): David A. Zidar

Regulation of Drug and Palatable Food Overconsumption by Similar Peptide Systems

Journal: Current Drug Abuse Reviews
Volume: 4 Issue: 3 Year: 2011 Page: 163-173
Author(s): Irene Morganstern, Jessica R. Barson, Sarah F. Leibowitz

The Histamine H3 Receptor as a Therapeutic Drug Target for Metabolic Disorders: Status, Challenges and Opportunities

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 1430-1446
Author(s): Jean-Marc Plancher

Editorial [Hot topic: G-Protein Coupled Receptors: Drug Targets of Key Importance (Guest Editors: Luca Piali and Christoph Boss)]

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 6 Year: 2011 Page: 608-608
Author(s): Luca Piali, Christoph Boss

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