Search Result "Inverse agonism"


Drugs that Act Through Membrane Receptors and Involve an Action of Inverse Agonism

Ebook: Young People’s Visions of the World

Volume: 1 Year: 2010
Author(s): Gabriel Barreda-Gomez, Rafael Rodriguez-Puertas
Doi: 10.2174/97816080515951100101

Third Generation Antipsychotic Drugs: Partial Agonism or Receptor Functional Selectivity?

Journal: Current Pharmaceutical Design
Volume: 16 Issue: 5 Year: 2010 Page: 488-501
Author(s): Richard B. Mailman, Vishakantha Murthy

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 8 Year: 2010 Page: 768-778
Author(s): Charles A. Lunn

High-Density Lipoprotein-Raising Strategies: Update 2010

Journal: Current Pharmaceutical Design
Volume: 16 Issue: 1 Year: 2010 Page: 1517-1530
Author(s): Frank Spillmann, Heinz-Peter Schultheiss, Carsten Tschope, Sophie Van Linthout

Novel Approaches in the Treatment of Antipsychotic-Induced Hyperprolactinemia:The Role of Partial Agonists of D2 Dopaminergic Receptors

Journal: Recent Patents on Endocrine, Metabolic & Immune Drug Discovery
Volume: 4 Issue: 3 Year: 2010 Page: 230-240
Author(s): Domenico De Berardis, Tiziano Acciavatti, Daniela Campanella, Nicola Serroni, Luigi Olivieri, Carla Ranalli, Viviana Marasco, Alessandro Carano, Marilde Cavuto, Giuseppe Di Iorio, Monica Piersanti, Francesco S. Moschetta, Massimo Di Giannantonio

GPR55, a Lysophosphatidylinositol Receptor with Cannabinoid Sensitivity?

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 8 Year: 2010 Page: 799-813
Author(s): Tapio Nevalainen, Andrew J. Irving

The Cannabinoid 2 Receptor as a Potential Therapeutic Target for Sepsis

Journal: Endocrine, Metabolic & Immune Disorders - Drug Targets
Volume: 10 Issue: 3 Year: 2010 Page: 224-234
Author(s): Kevin Richard Kasten, Johannes Tschop, Matthias Hans Tschop, Charles Curtis Caldwell

Understanding Functional Residues of the Cannabinoid CB1 Receptor for Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 10 Issue: 8 Year: 2010 Page: 779-798
Author(s): Joong-Youn Shim

Sequence and Structural Elements in the Mechanism of Function of Rhodopsin-Like Family of G Protein-Coupled-Receptors

Journal: Recent Patents on Endocrine, Metabolic & Immune Drug Discovery
Volume: 4 Issue: 3 Year: 2010 Page: 219-229
Author(s): James M. Wachira

High Content Screening of CXCR2-Dependent Signalling Pathways

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 13 Issue: 1 Year: 2010 Page: 3-15
Author(s): Michael Wolff, Simone Krede, Dorothea Haasen, Jorg Wiedenmann, G. Ulrich Nienhaus, Barbara Kistler, Franz Oswald, Ralf Heilker

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