Search Result "Hsp90 inhibitor assays"


Research Article

Improving the Hsp90 Inhibitors Containing 4-(2,4-Dihydroxyphenyl)-1,2,3-thiadiazole Scaffold: Synthesis, Affinity and Effect on Cancer Cells

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 11 Year: 2017 Page: 1593-1603
Author(s): Egidijus Kazlauskas,Algirdas Brukstus,Herkus Petrikas,Vilma Petrikaite,Inga Cikotiene,Daumantas Matulis

Review Article

Targeting Hsp90-Cdc37: A Promising Therapeutic Strategy by Inhibiting Hsp90 Chaperone Function

Journal: Current Drug Targets
Volume: 18 Issue: 13 Year: 2017 Page: 1572-1585
Author(s): Lei Wang,Li Li,Kai Gu,Xiao-Li Xu,Yuan Sun,Qi-Dong You

Review Article

Novobiocin Analogs as Potential Anticancer Agents

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 9 Year: 2017 Page: 728-733
Author(s): Angelika Dlugosz, Anna Janecka

Review Article

Preclinical and Clinical Studies of Chidamide (CS055/HBI-8000), An Orally Available Subtype-selective HDAC Inhibitor for Cancer Therapy

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 6 Year: 2017 Page: 802-812
Author(s): Shuai Gao,Xiaoyang Li,Jie Zang,Wenfang Xu,Yingjie Zhang

Review Article

Oncogene Expression Modulation in Cancer Cell Lines by DNA G-Quadruplex-Interactive Small Molecules

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 4 Year: 2017 Page: 4873-4904
Author(s): Ana Paula Francisco,Alexandra Paulo

Research Article

Synthesis of Phenol-derivatives and Biological Screening for Anticancer Activity

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 1 Year: 2017 Page: 1710-1720
Author(s): Anzhelika Karjalainen,Phuong Doan,Jerome G. Chandraseelan,Ossi Sandberg,Olli Yli-Harja,Nuno R. Candeias,Meenakshisundaram Kandhavelu

Review Article

Breast Cancer: Current Molecular Therapeutic Targets and New Players

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 2 Year: 2017 Page: 152-163
Author(s): Siddavaram Nagini

Review Article

Influenza A Virus Nucleoprotein: A Highly Conserved Multi-Functional Viral Protein as a Hot Antiviral Drug Target

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 20 Year: 2017 Page: 2271-2285
Author(s): Yanmei Hu,Hannah Sneyd,Raphael Dekant,Jun Wang

Review Article

Small-molecule Modulation of HDAC6 Activity: The Propitious Therapeutic Strategy to Vanquish Neurodegenerative Disorders

Journal: Current Medicinal Chemistry
Volume: 24 Issue: 37 Year: 2017 Page: 4104-4120
Author(s): Shabir A. Ganai

Review Article

Implications of Epigenetic Mechanisms and their Targets in Cerebral Ischemia Models

Journal: Current Neuropharmacology
Volume: 15 Issue: 6 Year: 2017 Page: 815-830
Author(s): Priya Jhelum,Bhanu C. Karisetty,Arvind Kumar,Sumana Chakravarty

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