Search Result "Hsp90 inhibitor assays"


Inhibitor Binding to Hsp90: A Review of Thermodynamic, Kinetic, Enzymatic, and Cellular Assays

Journal: Current Protein & Peptide Science
Volume: 15 Issue: 3 Year: 2014 Page: 256-282
Author(s): Vilma Petrikait e, Daumantas Matulis

HSP90 Inhibitors: Current Development and Potential in Cancer Therapy

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 9 Issue: 1 Year: 2014 Page: 1-20
Author(s): Katerina Sidera,Evangelia Patsavoudi

Synthesis and Evaluation of 4-arylmethyl Curcumin Analgues as Potent Hsp90 Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 8 Year: 2014 Page: 993-999
Author(s): Yang Liu,Min Ye,Qundan Wu,Lixian Wu,Jianhua Xu

IL-6 Activated JAK/STAT3 Pathway and Sensitivity to Hsp90 Inhibitors in Multiple Myeloma

Journal: Current Medicinal Chemistry
Volume: 21 Issue: 26 Year: 2014 Page: 3042-3047
Author(s): I. Kolosenko,D. Grander,K.P. Tamm

Antiproliferative Effect of HSP90 Inhibitor Y306zh Against Pancreatic Cancer is Mediated by Interruption of AKT and MAPK Signaling Pathways

Journal: Current Cancer Drug Targets
Volume: 14 Issue: 7 Year: 2014 Page: 671-683
Author(s): Nina Xue,Jing Jin,Di Liu,Rui Yan,Sen Zhang,Xiaoming Yu,Xiaoguang Chen

Protozoan HSP90-Heterocomplex: Molecular Interaction Network and Biological Significance

Journal: Current Protein & Peptide Science
Volume: 15 Issue: 3 Year: 2014 Page: 245-255
Author(s): Maria J. Figueras, Pablo C. Echeverria, Sergio O. Angel

Virtual Screening and Molecular Descriptor Analysis on Dietary Phytochemicals Against Heat Shock Protein 90 Enzyme

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 1 Year: 2014 Page: 40-49
Author(s): Salam Pradeep Singh,Bolin Kumar Konwar

Progress of HDAC Inhibitor Panobinostat in the Treatment of Cancer

Journal: Current Drug Targets
Volume: 15 Issue: 6 Year: 2014 Page: 622-634
Author(s): Xiaoyang Li,Jian Zhang,Yuanchao Xie,Yuqi Jiang,Zhang Yingjie,Wenfang Xu

Antitumor Effects of Celastrol and Semi-Synthetic Derivatives

Journal: Mini-Reviews in Organic Chemistry
Volume: 11 Issue: 3 Year: 2014 Page: 400-407
Author(s): Jorge A.R. Salvador,Rita C. Santos,Sandra A.C. Figueiredo,Yongkui Jing

Signaling Pathways Modulating Dependence of Lung Cancer on Mutant Epidermal Growth Factor Receptor and Mechanisms of Intrinsic and Acquired Resistance to Tyrosine Kinase Inhibitors

Journal: Current Pharmaceutical Design
Volume: 20 Issue: 24 Year: 2014 Page: 3883-3893
Author(s): Luciano Wannesson,Santiago Viteri,Carlota Costa,Niki Karachaliou,Miguel Angel Molina-Vila,Rafael Rosell

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