Search Result "HBA."


Research Article

Development of Novel Selective Pharmacophore for Tankyrase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 10 Year: 2017 Page: 1164-1175
Author(s): Xin Qiao,Ting Ran,Yan-Min Zhang,Jing Pan,Ling-Feng Yin,Wei-Neng Zhou,Lu Zhu,Jun-Nan Zhao,Hai-Chun Liu,Shuai Lu,Tao Lu,Ya-Dong Chen,Yu-Lei Jiang

Research Article

3D-QSAR Studies of HDAC6 Inhibitors Using Docking-Based Alignment

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 7 Year: 2017 Page: 798-810
Author(s): Chunqi Hu, Liang Hong, Jun Li, Wenting Du

Research Article

Surrogates of Insulin Sensitivity and Indices of Cardiometabolic Profile in Obesity

Journal: Current Vascular Pharmacology
Volume: 15 Issue: 4 Year: 2017 Page: 380-389
Author(s): Djordje S. Popovic, Edita Stokic, Milena Mitrovic, Dragana Tomic-Naglic, Radoslav Pejin, Tijana Icin, Bojan Vukovic, Zeljko Zivanovic, Sladjana Pejakovic, Branka Kovacev-Zavisic

Research Article

Advanced Structure-activity Relationships Applied to Mentha spicata L. Subsp. spicata Essential Oil Compounds as AChE and NMDA Ligands, in Comparison with Donepezil, Galantamine and Memantine – New Approach in Brain Disorders Pharmacology

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 16 Issue: 7 Year: 2017 Page: 800-811
Author(s): Speranta Avram,Maria Mernea,Eyup Bagci,Lucian Hritcu,Livia-Cristina Borcan,Dan Florin Mihailescu

Research Article

In Silico Modeling for the Design of 2-substitted Benzimidazole Derivatives, and Prediction of Activity as Procaspase-3 Activators and Apoptosis Inducer

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 4 Year: 2017 Page: 387-397
Author(s): Prajakta U. Kulkarni,Manjunath D. Ghate,Vivek K. Vyas

Review Article

SGLT-2 Inhibitors and Cardiovascular Risk in Diabetes Mellitus: A Comprehensive and Critical Review of the Literature

Journal: Current Pharmaceutical Design
Volume: 23 Issue: 1 Year: 2017 Page: 1510-1521
Author(s): Konstantinos Imprialos,Charles Faselis,Chrysoula Boutari,Konstantinos Stavropoulos,Vasilios Athyros,Asterios Karagiannis,Michael Doumas

Research Article

Quantification of Specific Glycation Sites in Human Serum Albumin as Prospective Type 2 Diabetes Mellitus Biomarkers

Journal: Protein & Peptide Letters
Volume: 24 Issue: 1 Year: 2017 Page: 887-896
Author(s): Sandro Spiller,Andrej Frolov,Ralf Hoffmann

Research Article

1,2,3-Triazole-Isoxazole Based Acetylcholinesterase Inhibitors: Synthesis, Biological Evaluation and Docking Study

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 1 Year: 2017 Page: 58-65
Author(s): Zahra Najafi,Mohammad Mahdavi,Mina Saeedi,Reyhaneh Sabourian,Mahnaz Khanavi,Maliheh Safavi,Maliheh Barazandeh Tehrani,Abbas Shafiee,Alireza Foroumadi,Tahmineh Akbarzadeh

Review Article

Current State and Future Perspectives in QSAR Models to Predict Blood- Brain Barrier Penetration in Central Nervous System Drug R&D

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 247-257
Author(s): Juan F. Morales,Sebastian Scioli Montoto,Pietro Fagiolino,Maria E. Ruiz

Research Article

Default Mode Network Connectivity and Related White Matter Disruption in Type 2 Diabetes Mellitus Patients Concurrent with Amnestic Mild Cognitive Impairment

Journal: Current Alzheimer Research
Volume: 14 Issue: 11 Year: 2017 Page: 1238-1246
Author(s): Di Qi,Ailin Wang,Yaojing Chen,Kewei Chen,Sisi Zhang,Junying Zhang,Xin Li,Lin Ai,Zhanjun Zhang

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