Search Result "Enzyme inhibition"


Research Article

Inhibition of Butyrylcholinesterase with Fluorobenzylcymserine, An Experimental Alzheimer's Drug Candidate: Validation of Enzoinformatics Results by Classical and Innovative Enzyme Kinetic Analyses

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 16 Issue: 7 Year: 2017 Page: 820-827
Author(s): Mohammad A. Kamal,Shazi Shakil,Muhammad S. Nawaz,Qian-sheng Yu,David Tweedie,Y. Tan,Xianqin Qu,Nigel H. Greig

Research Article

Inhibition of Product Template (PT) Domain of Aflatoxin Producing Polyketide Synthase Enzyme of Aspergillus parasiticus

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 7 Year: 2017 Page: 811-818
Author(s): Maneesh Kumar, Sindhuprava Rana, Harish Kumar, Jainendra Kumar, Rani Mansuri, Ganesh Chandra Sahoo

Review Article

Xanthine Oxidase and its Role as Target in Cardiovascular Disease: Cardiovascular Protection by Enzyme Inhibition?

Journal: Current Pharmaceutical Design
Volume: 23 Issue: 23 Year: 2017 Page: 3391-3404
Author(s): Mirjam Schuchardt,Jaqueline Herrmann,Markus Tolle,Markus van der Giet

Research Article

Quantitative In Silico Analysis of D-Amino Acid Oxidase Reactivity and Inhibition

Journal: Current Bioactive Compounds
Volume: 13 Issue: 4 Year: 2017 Page: 312-317
Author(s): Toshihiko Hanai

Research Article

The Effects of Drug Metabolizing Enzyme Inhibitors on Hepatic Efflux and Uptake Transporters

Journal: Drug Metabolism Letters
Volume: 11 Issue: 2 Year: 2017 Page: 111-118
Author(s): Jonathan Cheong,Jason S. Halladay,Emile Plise,Jasleen K. Sodhi,Laurent Salphati

Review Article

Pharmacokinetics of Gefitinib: Roles of Drug Metabolizing Enzymes and Transporters

Journal: Current Drug Delivery
Volume: 14 Issue: 2 Year: 2017 Page: 282-288
Author(s): Can Zhao,Shu-Yan Han,Ping-Ping Li

Review Article

Liposomal Encapsulation Enzymes: From Medical Applications to Kinetic Characteristics

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 17 Issue: 4 Year: 2017 Page: 366-370
Author(s): M. Jahadi,K. Khosravi-Darani

Review Article

Endogenous Biomarkers to Assess Drug-Drug Interactions by Drug Transporters and Enzymes

Journal: Current Drug Metabolism
Volume: 18 Issue: 8 Year: 2017 Page: 757-768
Author(s): T. Thanga Mariappan,Hong Shen,Punit Marathe

Review Article

The Role of Metabolizing Enzymes and Transporters in Antiretroviral Therapy

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 340-360
Author(s): Ling Ye,Chuqi Hou,Shuwen Liu

Review Article

Applying Knowledge of Enzyme Biochemistry to the Prediction of Functional Sites for Aiding Drug Discovery

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 21 Year: 2017 Page: 2401-2421
Author(s): Priyadarshini P. Pai,Sukanta Mondal

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