Search Result "EGFR-TKI resistance"


Overcoming Resistance to EGFR Inhibitors in NSCLC

Journal: Reviews on Recent Clinical Trials
Volume: 11 Issue: 2 Year: 2016 Page: 99-105
Author(s): Paolo Maione, Paola C. Sacco, Francesca Casaluce, Assunta Sgambato, Giuseppe Santabarbara, Antonio Rossi, Cesare Gridelli

Research Article

4-Anilinoquinazoline Derivatives with Epidermal Growth Factor Receptor Inhibitor Activity

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 12 Year: 2016 Page: 1652-1664
Author(s): Fang Liu,Baoding Tang,Hao Liu,Leina Li,Gang Liu,Yun Cheng,Yan Xu,Wenwen Chen,Yinjiu Huang

Review Article

Development of the Third Generation EGFR Tyrosine Kinase Inhibitors for Anticancer Therapy

Journal: Current Medicinal Chemistry
Volume: 23 Issue: 2 Year: 2016 Page: 3343-3359
Author(s): Weiyan Cheng, Jianhua Zhou, Xin Tian, Xiaojian Zhang

Review Article

EGFR and EML4-ALK Updated Therapies in Non-Small Cell Lung Cancer

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 11 Issue: 4 Year: 2016 Page: 393-400
Author(s): Ramon Andrade De Mello,Davi J. J. Liu,Pedro N. Aguiar,Hakaru Tadokoro

Review Article

ABC Transporters in the Development of Multidrug Resistance in Cancer Therapy

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 3 Year: 2016 Page: 4705-4716
Author(s): Angelika Dlugosz, Anna Janecka

Targeting the Bone Microenvironment in Metastatic Castration-Resistant Prostate Cancer

Journal: Current Drug Targets
Volume: 17 Issue: 3 Year: 2016 Page: 276-289
Author(s): Pavlos Msaouel,Jose Nahun Galeas,Alejandro Recio Boiles,Ramiro Rancier Ruiz,Michael Koutsilieris

Pyrazolopyrimidine Derivatives as Antineoplastic Agents: with a Special Focus on Thyroid Cancer

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 86-93
Author(s): Silvia Martina Ferrari,Concettina La Motta,Stefania Sartini,Enke Baldini,Gabriele Materazzi,Ugo Politti,Ilaria Ruffilli,Salvatore Ulisse,Paolo Miccoli,Alessandro Antonelli,Poupak Fallahi

Review Article

Design Strategies, Structures and Molecular Interactions of Small Molecule Src Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 16 Issue: 8 Year: 2016 Page: 992-1002
Author(s): Sureyya Olgen

Review Article

MicroRNA as Regulators of Cancer Stem Cells and Chemoresistance in Colorectal Cancer

Journal: Current Cancer Drug Targets
Volume: 16 Issue: 9 Year: 2016 Page: 738-754
Author(s): Xiaoming Liu, Qi Fu, Yong Du, Yinxue Yang, William C. Cho

Review Article

Challenges and Strategies in Precision Medicine for Non-Small-Cell Lung Cancer

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 2 Year: 2016 Page: 4374-4385
Author(s): Joseph J. Sacco, Hussein Al-Akhrass, Cornelia M. Wilson

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