Search Result "EGFR inhibition"


Recent Advances in Small Molecule Inhibitors of VEGFR and EGFR Signaling Pathways

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 1571-1590
Author(s): Haizhen Zhong, J. Phillip Bowen

A Role for SNX1 in the Regulation of EGF-Dependent Phosphorylated EGFR Endocytosis Via the Early/Late Endocytic Pathway in a Gefitinib-Sensitive Human Lung Cancer Cells

Journal: Current Signal Transduction Therapy
Volume: 6 Issue: 3 Year: 2011 Page: 383-395
Author(s): Yukio Nishimura, Kiyoko Yoshioka, Soichi Takiguchi, Biborka Bereczky, Yusaku Nakabeppu, Kazuyuki Itoh

Predicting Efficacy and Toxicity in the Era of Targeted Therapy: Focus on Anti-EGFR and Anti-VEGF Molecules

Journal: Current Drug Metabolism
Volume: 12 Issue: 1 Year: 2011 Page: 944-955
Author(s): Michele Caraglia, Daniele Santini, Giuseppe Bronte, Sergio Rizzo, Giovanni Sortino, Giovam Battista Rini, Gaetana Di Fede, Antonio Russo

Epidermal Growth Factor Receptor Irreversible Inhibitors: Chemical Exploration of the Cysteine-Trap Portion

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 1019-1030
Author(s): C. Carmi, A. Lodola, S. Rivara, F. Vacondio, A. Cavazzoni, R. R. Alfieri, A. Ardizzoni, P. G. Petronini, M. Mor

Erlotinib in Glioblastoma - Lost in Translation?

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 11 Issue: 8 Year: 2011 Page: 748-755
Author(s): Georg Karpel-Massler, M. Andrew Westhoff, Richard E. Kast, Christian Rainer Wirtz, Marc-Eric Halatsch

HGF-MET in Resistance to EGFR Tyrosine Kinase Inhibitors in Lung Cancer

Journal: Current Signal Transduction Therapy
Volume: 6 Issue: 2 Year: 2011 Page: 228-233
Author(s): Seiji Yano, Wei Wang, Qi Li, Tadaaki Yamada, Shinji Takeuchi, Kunio Matsumoto, Yasuhiko Nishioka, Saburo Sone

Mechanisms of Acquired Resistance to Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitors and New Therapeutic Perspectives in Non Small Cell Lung Cancer

Journal: Current Drug Targets
Volume: 12 Issue: 6 Year: 2011 Page: 922-933
Author(s): Laura Bonanno, Antonio Jirillo, Adolfo Favaretto

Mechanisms of Resistance to Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitors in Patients with Advanced Non-Small-Cell Lung Cancer: Clinical and Molecular Considerations

Journal: Current Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2011 Page: 1613-1628
Author(s): A. Pallis, E. Briasoulis, H. Linardou, C. Papadimitriou, D. Bafaloukos, P. Kosmidis, S. Murray

Dasatinib: An Anti-Tumour Agent via Src Inhibition

Journal: Current Drug Targets
Volume: 12 Issue: 4 Year: 2011 Page: 563-578
Author(s): Antonio Gnoni, Ilaria Marech, Nicola Silvestris, Angelo Vacca, Vito Lorusso

Targeting ErbB Receptors in High-Grade Glioma

Journal: Current Pharmaceutical Design
Volume: 17 Issue: 2 Year: 2011 Page: 2468-2487
Author(s): Sabina Berezowska, Jurgen Schlegel

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