Search Result "DNA gyrase"


Anti-Mycobacterial Activity of Quinolones. Triazoloquinolones a New Class of Potent Anti-Mycobacterial Agents

Journal: Anti-Infective Agents in Medicinal Chemistry
Volume: 7 Issue: 2 Year: 2008 Page: 134-147
Author(s): Antonio Carta, Sandra Piras, Michele Palomba, Daniela Jabes, Paola Molicotti, Stefania Zanetti

Characterizing the Bi-Subunit Type IB DNA Topoisomerase of Leishmania Parasites; a Novel Scenario for Drug Intervention in Trypanosomatids

Journal: Current Drug Targets
Volume: 9 Issue: 1 Year: 2008 Page: 966-978
Author(s): Rosa M. Reguera, Rosario Diaz-Gonzalez, Yolanda Perez-Pertejo, Rafael Balana-Fouce

Kinetoplast as a Potential Chemotherapeutic Target of Trypanosomatids

Journal: Current Pharmaceutical Design
Volume: 14 Issue: 9 Year: 2008 Page: 847-854
Author(s): Maria Cristina Machado Motta

Synthesis, Antimycobacterial Activities and Phototoxic Evaluation of 5H-thiazolo[3,2-a]quinoline-4-carboxylic Acid Derivatives

Journal: Medicinal Chemistry
Volume: 4 Issue: 5 Year: 2008 Page: 482-491
Author(s): Murugesan Dinakaran, Palaniappan Senthilkumar, Perumal Yogeeswari, Arnab China, Valakunja Nagaraja, Dharmarajan Sriram

Combinatorial Biosynthesis, Metabolic Engineering and Mutasynthesis for the Generation of New Aminocoumarin Antibiotics

Journal: Current Topics in Medicinal Chemistry
Volume: 8 Issue: 8 Year: 2008 Page: 667-679
Author(s): L. Heide, B. Gust, C. Anderle, S.-M. Li

Targeting the Transcriptional and Translational Machinery of the Endosymbiotic Organelle in Apicomplexans

Journal: Current Drug Targets
Volume: 9 Issue: 1 Year: 2008 Page: 948-956
Author(s): Tobias Fleige, Dominique Soldati-Favre

Human Leukemia and Lymphoma Cell Lines as Models and Resources

Journal: Current Medicinal Chemistry
Volume: 15 Issue: 4 Year: 2008 Page: 339-359
Author(s): Roderick A.F. MacLeod, Stefan Nagel, Michaela Scherr, Bjorn Schneider, Wilhelm G. Dirks, Cord C. Uphoff, Hilmar Quentmeier, Hans G. Drexler

Whos Winning the War? Molecular Mechanisms of Antibiotic Resistance in Helicobacter pylori

Journal: Current Drug Therapy
Volume: 3 Issue: 3 Year: 2008 Page: 190-203
Author(s): Kathleen R. Jones, Jeong-Heon Cha, D. Scott Merrell

Dimeric Approaches to Anti-Cancer Chemotherapeutics

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 8 Issue: 7 Year: 2008 Page: 807-816
Author(s): M. K. Hadden, B. S.J. Blagg

Structure-Activity Relationship Study of a Series of N-Substituted Piperazinyl-Fluoroquinolones as Anti-Helicobacter pylori Agents

Journal: Medicinal Chemistry
Volume: 4 Issue: 5 Year: 2008 Page: 498-502
Author(s): A. Foroumadi, M. Safavi, S. Emami, F. Siavoshi, S. Najjari, F. Safari, A. Shafiee

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