Search Result "Anti-leishmanial activity"


Research Article

Synthesis of New Cyclic Imides Derived From Safrole, Structure- and Ligand-based Approaches to Evaluate Potential New Multitarget Agents Against Species of Leishmania

Journal: Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2020 Page: 39-51
Author(s): José Alixandre de Sousa Luis,Normando Alexandre da Silva Costa,Cristiane Cosmo Silva Luis,Bruno Freitas Lira,Petrônio Filgueiras Athayde-Filho,Tatjana Keesen de Souza Lima,Juliana da Câmara Rocha,Luciana Scotti,Marcus Tullius Scotti

Research Article

Molecular Docking, Antioxidant, Anticancer and Antileishmanial Effects of Newly Synthesized Quinoline Derivatives

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 1516-1529
Author(s): Zoonish Malghani,Arif-Ullah Khan,Muhammad Faheem,Muhammad Z. Danish,Humaira Nadeem,Sameen F. Ansari,Madeeha Maqbool

Review Article

Thiocoumarins and Dithiocoumarins: Advances in Synthesis and Pharmacological Activity

Journal: Current Organic Chemistry
Volume: 24 Issue: 1 Year: 2020 Page: 1793-1814
Author(s): Diksha Chaudhary,Tanay Pramanik,Soumava Santra

Research Article

Synthesis and Biological Activity of Some Aminothiazole Derivatives as Antileishmanial Agents

Journal: Anti-Infective Agents
Volume: 18 Issue: 2 Year: 2020 Page: 178-189
Author(s): Zahra Rezaei,Bahador Sarkari,Soghra Khabnadideh,Mahbobeh Farjami,Mahsa Mehrjou,Atefeh Yazdi,Elham Riazimontazer,Mohammad Fararouei

Research Article

Biological Evaluation of 2-aminothiazole Hybrid as Antimalarial and Antitrypanosomal Agents: Design and Synthesis

Journal: Anti-Infective Agents
Volume: 18 Issue: 2 Year: 2020 Page: 101-108
Author(s): Surender S. Jadav,Vishnu N. Badavath,Ramesh Ganesan,Narayana M. Ganta,Dominique Besson,Venkatesan Jayaprakash

Research Article

Isolation, Characterization and Preliminary Cytotoxic and Antifungal Evaluations of Novel Lancifoliate Isolated from Methanol Extract of Conocarpus lancifolius

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 20 Issue: 1 Year: 2020 Page: 1664-1672
Author(s): Malik Saadullah,Muhammad Asif,Bashir A. Ch,Hafiza S. Yaseen,Muhammad Uzair,Khurram Afzal

Research Article

Revision of the Regioselectivity of the Beirut Reaction of Monosubstituted Benzofuroxans with Benzoylacetonitrile. 6-Substituted quinoxaline-2-carbonitrile 1,4- dioxides: Structural Characterization and Estimation of Anticancer Activity and Hypoxia Selectivity

Journal: Current Organic Synthesis
Volume: 17 Issue: 1 Year: 2020 Page: 29-39
Author(s): Galina I. Buravchenko,Alexander M. Scherbakov,Alexander А. Korlukov,Pavel V. Dorovatovskii,Andrey E. Shchekotikhin

Research Article

Transition Metal-free Approach for the Synthesis of 2-substituted Quinazolin-4(3H)-one via Anhydrous Magnesium Perchlorate

Journal: Current Organocatalysis
Volume: 7 Issue: 2 Year: 2020 Page: 118-123
Author(s): Shweta Mishra,Debashree Das,Adarsh Sahu,Shailendra Patil,Ram Kishor Agarwal,Asmita Gajbhiye

Review Article

Recent Advances in 1,3,5-Triazine Derivatives as Antibacterial Agents

Journal: Mini-Reviews in Organic Chemistry
Volume: 17 Issue: 8 Year: 2020 Page: 991-1041
Author(s): Divya Utreja,Jagdish Kaur,Komalpreet Kaur,Palak Jain

Review Article

Recent Theoretical Studies Concerning Important Tropical Infections

Journal: Current Medicinal Chemistry
Volume: 27 Issue: 5 Year: 2020 Page: 795-834
Author(s): Marcus Tullius Scotti,Alex France Messias Monteiro,Jéssika de Oliveira Viana,Francisco Jaime Bezerra Mendonça Junior,Hamilton M. Ishiki,Ernestine Nkwengoua Tchouboun,Rodrigo Santos A. De Araújo,Luciana Scotti

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