Search Result "ATP-binding pocket"


Docking and Molecular Dynamics Study on the Inhibitory Activity of Novel Inhibitors on Epidermal Growth Factor Receptor (EGFR)

Journal: Medicinal Chemistry
Volume: 7 Issue: 1 Year: 2011 Page: 24-31
Author(s): Qing-Hua Liao, Qing-Zhi Gao, Jing Wei, Kuo-Chen Chou

Peptides Targeting Estrogen Receptor Alpha-Potential Applications for Breast Cancer Treatment

Journal: Current Pharmaceutical Design
Volume: 17 Issue: 2 Year: 2011 Page: 2632-2653
Author(s): Guy Leclercq, Dominique Gallo, Janine Cossy, Ioanna Laios, Denis Larsimont, Guy Laurent, Yves Jacquot

The Coordinated Role of CYP450 Enzymes and P-gp in Determining Cancer Resistance to Chemotherapy

Journal: Current Drug Metabolism
Volume: 12 Issue: 8 Year: 2011 Page: 713-721
Author(s): Amalia Azzariti, Letizia Porcelli, Anna Elisa Quatrale, Nicola Silvestris, Angelo Paradiso

Recent Developments in the Third Generation Inhibitors of Bcr-Abl for Overriding T315I Mutation

Journal: Current Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2011 Page: 2146-2157
Author(s): X. Y. Lu, Q. Cai, K. Ding

Peptides or Small Molecules? Different Approaches to Develop More Effective CDK Inhibitors

Journal: Current Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2011 Page: 2854-2866
Author(s): D. Cirillo, F. Pentimalli, A. Giordano

In silico Designing and Screening of Lead Compounds to NS5-Methyltransferase of Dengue Viruses

Journal: Medicinal Chemistry
Volume: 7 Issue: 6 Year: 2011 Page: 655-662
Author(s): Dakshinamurthy Sivakumar, Thirunavukkarasu Sivaraman

Editorial [Hot Topic: Current Research on Protein Kinases (Guest Editors: Jari Yli-Kauhaluoma & Raimo K. Tuominen)]

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 1304-1304
Author(s): Jari Yli-Kauhaluoma, Raimo K. Tuominen

Bacterial Eukaryotic Type Serine-Threonine Protein Kinases: From Structural Biology to Targeted Anti-Infective Drug Design

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 1352-1369
Author(s): Valery N. Danilenko, Dmitry I. Osolodkin, Sergey A. Lakatosh, Maria N. Preobrazhenskaya, Alexander A. Shtil

Developments in Selective Small Molecule ATP-Targeting the Serine/Threonine Kinase Akt/PKB

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 11 Issue: 1 Year: 2011 Page: 1093-1107
Author(s): P. Wang, L. Zhang, Q. Hao, G. Zhao

Protein Flexibility and Ligand Recognition: Challenges for Molecular Modeling

Journal: Current Topics in Medicinal Chemistry
Volume: 11 Issue: 2 Year: 2011 Page: 192-210
Author(s): Francesca Spyrakis, Axel BidonChanal, Xavier Barril, F. Javier Luque

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