Search Result "ADMET studies"


Research Article

Anticancer Activity and In Silico ADMET Properties of 2,4,5-Trisubstitutedthiazole Derivatives

Journal: Current Drug Metabolism
Volume: 22 Issue: 7 Year: 2021 Page: 532-536
Author(s): Bilal A. Al-Jaidi,Soha T. Telfah,Sanaa K. Bardaweel,Pran K. Deb,Pobitra Borah,Katharigatta N. Venugopala,Yazan A. Bataineh,Qutaiba A. Al Khames Aga

Mini-Review Article

A Recent Appraisal of Artificial Intelligence and in Silico ADMET Prediction in the Early Stages of Drug Discovery

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 21 Issue: 1 Year: 2021 Page: 2786-2798
Author(s): Avinash Kumar,Suvarna G Kini,Ekta Rathi

Research Article

Molecular Docking, DFT Studies and ADMET Simulations for Evaluating Already Approved FDA Drugs as Inhibitors for SARS-Cov-2 RNADependent Polymerase

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 7 Year: 2021 Page: 674-685
Author(s): Manos C. Vlasiou,Kyriakos I. Ioannou,Kyriaki S. Pafiti

Research Article

Detection of Natural Inhibitors against Human Liver Cancer Cell Lines through QSAR, Molecular Docking and ADMET Studies

Journal: Current Topics in Medicinal Chemistry
Volume: 21 Issue: 8 Year: 2021 Page: 686-695
Author(s): Sarfaraz Alam,Sadaf Nasreen,Ateeque Ahmad,Mahendra Pandurang Darokar,Feroz Khan

Research Article

Analysis of Inhibitor Binding Combined with Reactivity Studies to Discover the Potentially Inhibiting Phytochemicals Targeting Chikungunya Viral Replication

Journal: Current Drug Discovery Technologies
Volume: 18 Issue: 3 Year: 2021 Page: 437-450
Author(s): Nouman Rasool,Afreen Bakht,Waqar Hussain

Research Article

Pharmacophore-based screening for identification of Human Acyl-CoA cholesterol acyltransferase inhibitors: An in-silico study

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 0 Year: 2021 Page: 1-14
Author(s): Shasta Kalra,Puja Kumari,Ankit Dhaundiyal

Research Article

In vitro, in vivo and in silico Antihyperglycemic Activity of Some Semi-synthetic Phytol Derivatives

Journal: Medicinal Chemistry
Volume: 17 Issue: 0 Year: 2021 Page: 1-7
Author(s): Harish C. Upadhyay,Akansha Mishra,Jyotsana Pandey,Pooja Sharma,Akhilesh K. Tamrakar,Arvind K. Srivastava,Feroz Khan,Santosh K. Srivastava

Research Article

In-silico Studies and Wet-Lab Validation of Camptothecin Derivatives for Anti-Cancer Activity Against Liver (HepG2) and Lung (A549) Cancer Cell Lines

Journal: Current Topics in Medicinal Chemistry
Volume: 21 Issue: 1 Year: 2021 Page: 908-919
Author(s): Komal Kalani,Dharmendra K. Yadav,Sarfaraz Alam,Feroz Khan,Mahendra P. Kashyap,Santosh K. Srivastava,Aditya B. Pant

Research Article

Synthesis of Novel Aryl (4-Aryl-1h-Pyrrol-3-Yl) (Thiophen-2-Yl) Methanone Derivatives: Molecular Modelling, In Silico Admet, Anti-Inflammatory and Anti-Ulcer Activities

Journal: Anti-Inflammatory & Anti-Allergy Agents in Medicinal Chemistry
Volume: 20 Issue: 2 Year: 2021 Page: 182-195
Author(s): Arif Pasha,Sumanta Mondal,Naresh Panigrahi

Research Article

Analyzing Phytochemicals as Inhibitors of Diabetes Mellitus 2 Causing Proteins based on Computer-Aided Drug Discovery Protocols

Journal: The Natural Products Journal
Volume: 11 Issue: 3 Year: 2021 Page: 383-391
Author(s): Sobia Nazir Chaudry,Waqar Hussain,Nouman Rasool

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