Search Result "ADMET score"


Research Article

In-silico Design, ADMET Screening, MM-GBSA Binding Free Energy of Some Novel Isoxazole Substituted 9-anilinoacridines as HER2 Inhibitors Targeting Breast Cancer

Journal: Current Drug Research Reviews
Volume: 11 Issue: 2 Year: 2019 Page: 118-128
Author(s): Rajagopal Kalirajan,Arumugasamy Pandiselvi,Byran Gowramma,Pandiyan Balachandran

Research Article

In-silico Designing, ADMET Analysis, Synthesis and Biological Evaluation of Novel Derivatives of Diosmin Against Urease Protein and Helicobacter pylori Bacterium

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2019 Page: 2658-2675
Author(s): Ritu Kataria,Anurag Khatkar

Research Article

2,4-Dichloro-5-[(N-aryl/alkyl)sulfamoyl]benzoic Acid Derivatives: In Vitro Antidiabetic Activity, Molecular Modeling and In silico ADMET Screening

Journal: Medicinal Chemistry
Volume: 15 Issue: 2 Year: 2019 Page: 186-195
Author(s): Samridhi Thakral,Vikramjeet Singh

Research Article

Ligand-Based Pharmacophore Modeling and Virtual Screening to Discover Novel CYP1A1 Inhibitors

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 2782-2794
Author(s): Rana Adnan Tahir,Farwa Hassan,Abdul Kareem,Umer Iftikhar,Sheikh Arslan Sehgal

Research Article

A Computer - Aided Drug Designing for Pharmacological Inhibition of Mutant ALK for the Treatment of Non-small Cell Lung Cancer

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 1129-1144
Author(s): Saphy Sharda,Ravina Khandelwal,Ritu Adhikary,Diksha Sharma,Manisha Majhi,Tajamul Hussain,Anuraj Nayarisseri,Sanjeev Kumar Singh

Research Article

Search for Potential Inducible Nitric Oxide Synthase Inhibitors with Favorable ADMET Profiles for the Therapy of Helicobacter pylori Infections

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 2795-2804
Author(s): Ricardo Pereira Rodrigues,Juliana Santa Ardisson,Rita de Cássia Ribeiro Gonçalves,Tiago Branquinho Oliveira,Vinicius Barreto da Silva,Daniel Fábio Kawano,Rodrigo Rezende Kitagawa

Research Article

Pharmacophore Modeling, Synthesis, Scaffold Hopping and Biological β- Hematin Inhibition Interaction Studies for Anti-malaria Compounds

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 2743-2765
Author(s): Neda Fayyazi,Somayeh Esmaeili,Salman Taheri,Frederico F. Ribeiro,Marcus T. Scotti,Luciana Scotti,Jahan B. Ghasemi,Lotfollah Saghaei,Afshin Fassihi

Research Article

Antiangiogenesis Potential of Alpinumisoflavone as an Inhibitor of Matrix Metalloproteinase-9 (MMP-9) and Vascular Endothelial Growth Factor Receptor-2 (VEGFR-2)

Journal: Current Enzyme Inhibition
Volume: 15 Issue: 3 Year: 2019 Page: 159-178
Author(s): Honeymae C. Alos,Junie B. Billones,Ross D. Vasquez,Agnes L. Castillo

Research Article

Synthesis, Biological Evaluation and Molecular Docking Studies of Novel Di-hydropyridine Analogs as Potent Antioxidants

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 2 Year: 2019 Page: 2676-2686
Author(s): Saddala Madhu Sudhana,Pradeepkiran Jangampalli Adi

Research Article

Identification of High-affinity Small Molecules Targeting Gamma Secretase for the Treatment of Alzheimer’s Disease

Journal: Current Topics in Medicinal Chemistry
Volume: 19 Issue: 1 Year: 2019 Page: 1173-1187
Author(s): Meer Asif Ali,Sugunakar Vuree,Himshikha Goud,Tajamul Hussain,Anuraj Nayarisseri,Sanjeev Kumar Singh

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