Search Result "ADMET score"


Research Article

Molecular Docking, In-Silico ADMET Study and Development of 1,6- Dihydropyrimidine Derivative as Protein Tyrosine Phosphatase Inhibitor: An Approach to Design and Develop Antidiabetic Agents

Journal: Current Computer-Aided Drug Design
Volume: 14 Issue: 4 Year: 2018 Page: 349-362
Author(s): Ashish D. Patel,Rahul Barot,Inaxi Parmar,Ishan Panchal,Umang Shah,Mehul Patel,Bharat Mishtry

Research Article

Structure-based Virtual Screening for the Identification of High-affinity Small Molecule Towards STAT3 for the Clinical Treatment of Osteosarcoma

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 2 Year: 2018 Page: 2511-2526
Author(s): Ravina Khandelwal,Aashish Pratap Singh Chauhan,Swarnima Bilawat,Aishwarya Gandhe,Tajamul Hussain,Elizabeth Anne Hood,Anuraj Nayarisseri,Sanjeev Kumar Singh

Research Article

Virtual Screening of Novel Glucosamine-6-Phosphate Synthase Inhibitors

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 21 Issue: 3 Year: 2018 Page: 182-193
Author(s): Amit Lather,Sunil Sharma,Anurag Khatkar

Research Article

High Throughput Screening Based Highly Potent Sulfonylbenzamide Anti-diabetic Drug

Journal: Current Drug Therapy
Volume: 13 Issue: 2 Year: 2018 Page: 162-173
Author(s): Sayantan Pradhan,Chittaranjan Sinha

Research Article

In Silico Bioactivity Prediction of Methoxime-3,4-dephostatin Derivatives on Human PTP1B: Search for Novel Antidiabetic Leads

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 5 Year: 2018 Page: 500-507
Author(s): Sabina B. Choudhury,Anupam D. Talukdar,Manabendra D. Choudhury,Monjur A. Laskar,Abhishek Chowdhury

Research Article

In silico Structure-based Identification of Novel Acetylcholinesterase Inhibitors Against Alzheimer’s Disease

Journal: CNS & Neurological Disorders - Drug Targets
Volume: 17 Issue: 1 Year: 2018 Page: 54-68
Author(s): Kanzal Iman,Muhammad Usman Mirza,Nauman Mazhar,Michiel Vanmeert,Imran Irshad,Mohammad A. Kamal

Research Article

QSAR and Molecular Docking Studies on a Series of 1-Amino-5H-pyrido [4, 3-b]indol-4-carboxamides Acting as Janus Kinase 2 (JAK2) Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 2 Year: 2018 Page: 169-180
Author(s): Basheerulla Shaik,Satya P. Gupta,Tabassum Zafar,K. Anita

Research Article

A Therapeutic Paradigm to Appraise the Competence of Chitosan Oligosaccharide Lactate Targeting Monoamine Oxidase-A and PGlycoprotein to Contest Depression by Channeling the Blood Brain Barrier

Journal: Current Bioinformatics
Volume: 13 Issue: 3 Year: 2018 Page: 273-279
Author(s): A. Anita Margret,Ganesh Kumar Arumugam

Research Article

Computer-aided Drug Designing for the Identification of High-Affinity Small Molecule Targeting CD20 for the Clinical Treatment of Chronic Lymphocytic Leukemia (CLL)

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 2 Year: 2018 Page: 2527-2542
Author(s): Tajamul Hussain,Kritika Sinha,Manisha Majhi,Garima Thakur,Khushboo Patidar,Jajoriya Sweta,Anuraj Nayarisseri,Sanjeev Kumar Singh

Research Article

An In Silico Investigation of Potential EGFR Inhibitors for the Clinical Treatment of Colorectal Cancer

Journal: Current Topics in Medicinal Chemistry
Volume: 18 Issue: 2 Year: 2018 Page: 2338-2349
Author(s): Manisha Majhi,Meer Asif Ali,Akanksha Limaye,Kritika Sinha,Praveena Bairagi,Megha Chouksey,Ruchi Sukhla,Tajamul Hussain,Nisha Kanwar,Anuraj Nayarisseri,Sanjeev Kumar Singh

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