Search Result "5-pyrazole derived ligands"


Research Article

Design, Synthesis and Biological Evaluation of 1-methyl-1H-pyrazole-5-Carboxamide Derivatives as Novel Anti-Prostate Cancer Agents

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 0 Year: 2021 Page: 1-11
Author(s): Xin Chen,Changqing Xu,Yuxia Li,Xiaoming Duan,Guisen Zhao

Research Article

Molecular Docking Studies of Glycyrrhetinic Acid Derivatives as Anti- Colorectal Cancer Agents

Journal: Current Computer-Aided Drug Design
Volume: 17 Issue: 3 Year: 2021 Page: 429-444
Author(s): Nam Q.H. Doan,Tuyen N. Truong,Phuong T.V. Nguyen

MAO Inhibitory Activity of 4, 5-Dihydro-1 HPyrazole Derivatives: A Platform To Design Novel Antidepressants

Ebook: Frontiers in Drug Design and Discovery

Volume: 10 Year: 2021
Author(s): Vishnu Nayak Badavath,Venkatesan Jayaprakash
Doi: 10.2174/97898114215631211001
General Review Article

Synthetic and Biological Attributes of Pyrimidine Derivatives: A Recent Update

Journal: Current Organic Synthesis
Volume: 18 Issue: 0 Year: 2021 Page: 1-36
Author(s): Meenu Devi,Shivangi Jaiswal,Sonika Jain,Navjeet Kaur,Jaya Dwivedi

Review Article

Recent Updates on Pyrazoline Derivatives as Promising Candidates for Neuropsychiatric and Neurodegenerative Disorders

Journal: Current Topics in Medicinal Chemistry
Volume: 21 Issue: 0 Year: 2021 Page: 1-20
Author(s): T. M. Rangarajan,Bijo Mathew

Research Article

Design, Synthesis, Computational and Biological Evaluation of Two New Series of 1, 3- and 1,6-dihydroxy Xanthone Derivatives as Selective COX-2 Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 0 Year: 2021 Page: 1-31
Author(s): Urvashee Gogoi,Aparoop Das,Manash Pratim Pathak,Pronobesh Chattopadhyay,Surabhi Johari

Review Article

Design of New Improved Curcumin Derivatives to Multi-targets of Cancer and Inflammation

Journal: Current Drug Targets
Volume: 22 Issue: 5 Year: 2021 Page: 573-589
Author(s): A. Harikrishnan,V. Veena,Sunali Khanna

Research Article

Design, Synthesis, Molecular Docking, and Anticancer Evaluation of Pyrazole Linked Pyrazoline Derivatives with Carbothioamide Tail as EGFR Kinase Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 21 Issue: 1 Year: 2021 Page: 42-60
Author(s): Farah Nawaz,Ozair Alam,Ahmad Perwez,Moshahid A. Rizvi,Mohd. Javed Naim,Nadeem Siddiqui,Jannat ul Firdaus,Shakilur Rahman,Mukund Jha,Aadil A. Sheikh

Research Article

Synthesis, Cytotoxicity Evaluation and Molecular Docking of Fluorine Containing Hexahydroquinoline-3-Carbonitrile Derivatives

Journal: Current Drug Discovery Technologies
Volume: 18 Issue: 0 Year: 2021 Page: 1-11
Author(s): Nishith Teraiya,Subhas Karki,Ashlesha Chauhan

Research Article

Synthesis, Design and Anti-inflammatory Activity of Novel 5-(Indol-3- yl)thiazolidinone Derivatives as COX-2 Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 18 Issue: 6 Year: 2021 Page: 525-541
Author(s): Saad R. Atta-Allah,Nasser S.M. Ismail,Ibrahim F. Nassar

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