Search Result "4- thiadiazole"


Research Article

In Silico Appraisal, Synthesis, Antibacterial Screening and DNA Cleavage for 1,2,5-thiadiazole Derivative

Journal: Current Computer-Aided Drug Design
Volume: 15 Issue: 5 Year: 2019 Page: 445-455
Author(s): Suraj N. Mali,Sudhir Sawant,Hemchandra K. Chaudhari,Mustapha C. Mandewale

Research Article

Synthesis and Antioxidant Activity of Novel 5-amino-2-alkyl/glycosylthio-1,3,4- thiadiazoles: Regioselective Alkylation and Glycosylation of the 5-amino-1,3,4- thiadiazole-2-thiol Scaffold

Journal: Current Organic Synthesis
Volume: 16 Issue: 5 Year: 2019 Page: 801-809
Author(s): El Sayed H. El Ashry,El Sayed Ramadan,Mohammed R. Amer,Yeldez El Kilany,Mohamed E. I. Badawy,Entsar I. Rabea

Research Article

Synthesis Under Microwave Irradiation and Molecular Docking of Some Novel Bioactive Thiadiazoles

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 5 Year: 2019 Page: 437-447
Author(s): Sobhi M. Gomha,Mastora M. Edress,Zeinab A. Muhammad,Hatem M. Gaber,Mohamed M. Amin,Islam K. Matar

Research Article

Synthesis, Antioxidant and Antiurease Activities of Some New 5,6- dichloro-2-(4-fluorobenzyl)-1H-benzimidazole Derivatives Containing Furan, Oxadiazole, Triazole and Thiadiazole Moieties

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 8 Year: 2019 Page: 939-947
Author(s): Hakan Bektas,Canan Albay,Emre Menteşe,Bahar Bilgin Sokmen,Zafer Kurt,Dilem Şen

Research Article

In silico Molecular Docking and ADME Studies of 1,3,4-thiadiazole Derivatives in Relation to in vitro PON1 Activity

Journal: Current Computer-Aided Drug Design
Volume: 15 Issue: 2 Year: 2019 Page: 136-144
Author(s): Belgin Sever,Kaan Kucukoglu,Hayrunnisa Nadaroglu,Mehlika Dilek Altıntop

Research Article

Synthesis, Antioxidant and Anti-inflammatory Activities of 5-((styrylsulfonyl) methyl)-1,3,4-Oxadiazol / Thiadiazol-2-amine Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 1 Year: 2019 Page: 1233-1247
Author(s): Gundala Sravya,Ummadi Nagarjuna,Venkatapuram Padmavathi,Galla Rajitha,Sakuri Chandi priya,Adivireddy Padmaja

Research Article

Synthesis and Characterization of Some New 1,3,4-thiadiazole Compounds Derived from 3,4-(Methylenedioxy)cinnamic Acid and their Antimicrobial Activities

Journal: Letters in Organic Chemistry
Volume: 16 Issue: 1 Year: 2019 Page: 825-836
Author(s): Halit Muğlu,Mahmut Gür,Maesm Ahmed Mohamed Ben Hsin,Nesrin Şener,Sevil Özkınalı,Osman Emre Özkan,İzzet Şener

Research Article

Synthesis and Docking Study of Novel 4-Thiazolidinone Derivatives as Anti-Gram-positive and Anti-H. pylori Agents

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 239-249
Author(s): Armin Khomami,Mohammadamin Rahimi,Arash Tabei,Parastoo Saniee,Arash Mahboubi,Alireza Foroumadi,Nasrin Nassiri Koopaei,Ali Almasirad

Research Article

Design, Synthesis and Biological Activity of Some 4, 5-Disubstituted-2, 4- Dihydro-3H-1, 2, 4- Triazole-3-Thione Derivatives

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 19 Issue: 3 Year: 2019 Page: 197-205
Author(s): Krishan Kumar Verma,Umesh Kumar Singh,Jainendra Jain

Research Article

Synthesis, Structure Elucidation and Biological Activities of Some Novel 4(3H)-Quinazolinones as Anti-Biofilm Agents

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 3 Year: 2019 Page: 313-321
Author(s): Sevda Türk,Sevgi Karakuş,Abdulilah Ece,Seyhan Ulusoy,Gülgün Bosgelmez-Tınaz

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