Search Result "3-b]quinolone"


The 4-Quinolone-3-Carboxylic Acid Motif as a Multivalent Scaffold in Medicinal Chemistry

Journal: Current Medicinal Chemistry
Volume: 16 Issue: 1 Year: 2009 Page: 1746-1767
Author(s): Claudia Mugnaini, Serena Pasquini, Federico Corelli

Quinolones: Action and Resistance Updated

Journal: Current Topics in Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2009 Page: 981-998
Author(s): Karl Drlica, Hiroshi Hiasa, Robert Kerns, Muhammad Malik, Arkady Mustaev, Xilin Zhao

QSAR Studies on 4-Quinolone Derivatives as High-Affinity Ligands at the Benzodiazepine Site of Brain GABAA Receptors

Journal: Medicinal Chemistry
Volume: 5 Issue: 4 Year: 2009 Page: 353-358
Author(s): Anand Gaurav, Mange R. Yadav, Rajani Giridhar, Vertika Gautam, Ranjit Singh

Efficacy of Fluoroquinolones Against Pathogenic Oral Bacteria

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 1 Year: 2009 Page: 1147-1158
Author(s): V. Nunez Otero, J. Limeres Posse, I. Tomas Carmona, P. Diz Dios

A Convenient Synthesis of 1-Alkyl-7-chloro-6-fluoro-3-nitro-4-quinolones

Journal: Letters in Organic Chemistry
Volume: 6 Issue: 6 Year: 2009 Page: 511-514
Author(s): Raed A. Al-Qawasmeh, Jalal A. Zahra, Monther A. Khanfar, Yusuf M. AL-Hiari, Mustafa M. El-Abadelah, Wolfgang Voelter

Antibacterial Activity of Lipophilic Fluoroquinolone Derivatives

Journal: Medicinal Chemistry
Volume: 5 Issue: 5 Year: 2009 Page: 419-421
Author(s): Camila G. de Almeida, Claudio G. Diniz, Vania L. Silva, Mauricio F. Saraiva, Mireille Le Hyaric, Mauro V. de Almeida

3-Hydroxy-2-phenyl-4(1H)-quinolinones as Promising Biologically Active Compounds

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 6 Year: 2009 Page: 696-702
Author(s): P. Hradil, J. Hlavac, M. Soural, M. Hajduch, M. Kolar, R. Vecerova

Synthesis, In Vitro Activities of (2-Cyclopropoxyphenyl)piperidine Derivatives for α1a and α1d Adrenergic Receptor Inhibitors

Journal: Medicinal Chemistry
Volume: 5 Issue: 1 Year: 2009 Page: 15-22
Author(s): Shengjian Li, George Chiu, Virginia L. Pulito, Jingchun Liu, Peter J. Connolly, Steven A. Middleton

Molecular Determinants of Fluoroquinolone Antibacterial Agents Pharmacokinetics

Journal: Current Clinical Pharmacology
Volume: 4 Issue: 3 Year: 2009 Page: 191-197
Author(s): Dominique Leveque, Francois Jehl

Mechanisms of Resistance: Useful Tool to Design Antibacterial Agents for Drug - Resistant Bacteria

Journal: Mini-Reviews in Medicinal Chemistry
Volume: 9 Issue: 2 Year: 2009 Page: 194-205
Author(s): J. K. Savjani, A. K. Gajjar, K. T. Savjani

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