Search Result "3-Triazole"


Research Article

2-((1H-1,2,3-triazol-1-yl)methyl)-3-phenylquinazolin-4(3H)-ones: Design, Synthesis and Evaluation as Anti-cancer Agents

Journal: Current Bioactive Compounds
Volume: 14 Issue: 3 Year: 2018 Page: 254-263
Author(s): Kamala K. Vasu,Hemantkumar D. Ingawale,Sneha R. Sagar,Jayesh A. Sharma,Dhaivat H. Pandya,Milee Agarwal

Research Article

QSAR Analysis of 6-Fluoro-3-(4H- 1,2,4-triazol-3-yl)quinolin-4(1H)-ones as Antileukemic Agents using Physicochemical and Alignment Independent Topological Based Descriptors

Journal: Letters in Organic Chemistry
Volume: 15 Issue: 7 Year: 2018 Page: 551-558
Author(s): Yan Wang,Qin Zhou,Li Wang,Jun-Jie Ma

Research Article

Facile Synthesis, Crystal Structure, DFT Calculation and Biological Activities of 4-(2-fluorophenyl)-3-(3-methoxybenzyl)-1H-1,2,4-triazol-5 (4H)-one (5)

Journal: Medicinal Chemistry
Volume: 14 Issue: 5 Year: 2018 Page: 451-459
Author(s): Muhammad Saleem,Muhammad Rafiq,Yeon Ki Jeong,Dae Won Cho,Chong-Hyeak Kim,Sung-Yum Seo,Chang-Shik Choi,Seong-Karp Hong,Ki-Hwan Lee

Research Article

Novel Hydroxamic Acids Incorporating 1-((1H-1,2,3-Triazol-4-yl)methyl)- 3-substituted-2-oxoindolines: Synthesis, Biological Evaluation and SAR Analysis

Journal: Medicinal Chemistry
Volume: 14 Issue: 8 Year: 2018 Page: 831-850
Author(s): Do T.M. Dung,Nguyen V. Huan,Do M. Cam,Dao C. Hieu,Pham-The Hai,Le-Thi-Thu Huong,Jisung Kim,Jeong E. Choi,Jong S. Kang,Sang-Bae Han,Nguyen-Hai Nam

Research Article

Synthesis of Novel 6-(1H-pyrazol-4-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles as Potential Antimicrobial Agents

Journal: Letters in Organic Chemistry
Volume: 15 Issue: 2 Year: 2018 Page: 92-98
Author(s): Rashmi Pundeer,Pooja Ranjan,Richa Prakash,Radhika Joshi

Research Article

Synthesis, Characterization and Antibacterial Activity of Some New 1,2,4- Triazole Schiff bases and 1,2,4-triazolo[3,4-b][1,3,4]thiadiazines

Journal: Letters in Organic Chemistry
Volume: 15 Issue: 7 Year: 2018 Page: 575-582
Author(s): Kooi-Mow Sim,Pei-Qie Chan,Xin-Lik Boo,Ker-Sin Heng,Kah-Whei Lye,Kah-Cheng Teo

Research Article

Synthesis, Characterization and Antibacterial Evaluation of some New 1,2,4-triazolo[3,4-b][1,3,4]thiadiazines as Potential Antibacterial Agents

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 7 Year: 2018 Page: 733-743
Author(s): Kooi-Mow Sim,Kah-Cheng Teo

Research Article

Synthesis and Cytotoxicity Evaluation of Novel Tricyclic Dihydropyrazolo [4,3-f][1,2,3]triazolo Diazepines

Journal: Letters in Drug Design & Discovery
Volume: 15 Issue: 1 Year: 2018 Page: 1020-1025
Author(s): Chiranjeevi Bingi,Ashok Kale,Yedla Poornachandra,Chityal Ganesh Kumar,Krishnaiah Atmakur

Research Article

Microwave Assisted Syntheses of 4-Amino-carane-3-ols from 3,4- Epoxycarane and Heterocyclic Amines

Journal: Current Microwave Chemistry
Volume: 5 Issue: 1 Year: 2018 Page: 54-61
Author(s): Alexander M. Agafoncev,Tatyana A. Shumilova,Alexey V. Tkachev

Research Article

One-Pot Synthesis of Triazolo-Heterolignans: Biological Evaluation and Molecular Docking Studies as Tubulin Inhibitors

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 18 Issue: 1 Year: 2018 Page: 1702-1710
Author(s): Raji Reddy Chada,Nilesh Sasane,Muppidi Subbarao,Reddi Rani Valleti,Jonnalagadda Vijaykumar,Bhukya Supriya,Surender Singh Jadav,Ramesh Ummanni

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