Search Result "2D QSAR"


Research Article

2D, 3D, G-QSAR and Docking Studies of Thiazolyl-pyrazoline Analogues as Potent (Epidermal Growth Factor Receptor-tyrosine Kinase) EGFR-TK Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 11 Year: 2017 Page: 1228-1238
Author(s): Ghodgaonkar Sunayana,Bhandari Shashikant,Waghulde Sandeep

Research Article

New Research for Quinazoline-2,4-diones as HPPD Inhibitors Based on 2D-MLR and 3D-QSAR Models

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 9 Year: 2017 Page: 748-759
Author(s): Ying Fu,Yi-Na Sun,Hai-Feng Cao,Ke-Han Yi,Li-Xia Zhao,Jia-Zhong Li,Fei Ye

Research Article

Combined Approach of QSAR and Docking Studies for the Design of Local Anaesthetic Agents

Journal: Combinatorial Chemistry & High Throughput Screening
Volume: 20 Issue: 3 Year: 2017 Page: 272-276
Author(s): Chunyan Zhang,Zhi Li,Jiahai Ma,Jing Zhang,Longming Zhang,Tao Li,Shijian Zheng

Research Article

Peptide Drugs QSAR Study Based on Topomer CoMFA

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 10 Year: 2017 Page: 1114-1121
Author(s): Jianbo Tong,Lingxiao Li,Kangnan Li,Min Bai

Research Article

Docking and QSAR Studies of Aryl-valproic Acid Derivatives to Identify Antiproliferative Agents Targeting the HDAC8

Journal: Anti-Cancer Agents in Medicinal Chemistry
Volume: 17 Issue: 7 Year: 2017 Page: 927-940
Author(s): Heidy Martínez-Pacheco,Guillermo Ramírez-Galicia,Midalia Vergara-Arias,Jurg Gertsch,Jonathan Manuel Fragoso-Vazquez,David Mendez-Luna,A. L. Abujamra,Cabrera-Perez Laura Cristina,Rosales-Hernandez Martha Cecilia,I Mendoza-Lujambio,Jose Correa-Basurto

Research Article

Integrating Multiple Receptor Conformation Docking and Multi Dimensional QSAR for Enhancing Accuracy of Binding Affinity Prediction

Journal: Current Computer-Aided Drug Design
Volume: 13 Issue: 2 Year: 2017 Page: 127-142
Author(s): Vangala Radhika,Hassan A. Jaraf,Sivan S. Kanth,Manga Vijjulatha

Research Article

Predicting Isoform-specific Binding Selectivities of Benzensulfonamides Using QSAR and 3D-QSAR

Journal: Current Computer-Aided Drug Design
Volume: 13 Issue: 1 Year: 2017 Page: 75-83
Author(s): Vytautas Ra skevi cius, Visvaldas Kairys

Research Article

3D QSAR Analysis on 2piperidinopiperidinethiadiazole Derivatives as Histamine H3 Receptor Inhibitors

Journal: Current Nanomedicine
Volume: 7 Issue: 1 Year: 2017 Page: 59-66
Author(s): Yogesh Vaishnav,Pranita Kashyap,Chanchal Deep Kaur

Review Article

Learning from Multiple Classifier Systems: Perspectives for Improving Decision Making of QSAR Models in Medicinal Chemistry

Journal: Current Topics in Medicinal Chemistry
Volume: 17 Issue: 3 Year: 2017 Page: 3269-3288
Author(s): Hai Pham-The,Nguyen-Hai Nam,Doan-Viet Nga,Dang Thanh Hai,Karel Dieguez-Santana,Yovani Marrero-Ponce,Juan A. Castillo-Garit,Gerardo M. Casanola-Martin,Huong Le-Thi-Thu

Research Article

Docking and QSAR Studies of 1,4-Dihydropyridine Derivatives as Anti- Cancer Agent

Journal: Recent Patents on Anti-Cancer Drug Discovery
Volume: 12 Issue: 2 Year: 2017 Page: 174-185
Author(s): Shirin Mollazadeh, Jamal Shamsara, Maryam Iman, Farzin Hadizadeh

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