Search Result "2-a]pyridines"


Synthesis and Biological Evaluation of New imidazo[1,2-a]pyridine Derivatives as Selective COX-2 Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 8 Year: 2016 Page: 793-799
Author(s): Mahsa Azami Movahed, Bahram Daraei, Afshin Zarghi

Research Article

Schiff Bases of Benzothiazol-2-ylamine and Thiazolo[5,4-b] pyridin-2-ylamine as Anticonvulsants: Synthesis, Characterization and Toxicity Profiling*

Journal: Central Nervous System Agents in Medicinal Chemistry
Volume: 16 Issue: 3 Year: 2016 Page: 240-248
Author(s): Rashmi Shukla, Ajeet P. Singh, Pankaj K. Sonar, Mudita Mishra, Shailendra K. Saraf

Synthesis and Evaluation of Compounds Containing 4-arylpiperazinyl Moieties Linked to a 2-(pyridin-3-yl)-1H-benzimidazole as p38 MAP Kinase Inhibitors

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 7 Year: 2016 Page: 691-696
Author(s): Mohamed Ashraf Ali, Hasnah Osman, Raju Suresh Kumar, Abdulrahman I. Almansour, Natarajan Arumugam, Vijay H. Masand, Theivendren Panneerselvam

Discovery and Optimization of 1-(4-chloro-3-(trifluoromethyl)- phenyl)-3-(2-(amino)pyridin-3-yl)ureas as Novel KDR Kinase Inhibitors

Journal: Medicinal Chemistry
Volume: 12 Issue: 4 Year: 2016 Page: 328-337
Author(s): Yu Jiao,Fei Huang,Pengfei Xu,Yanmin Zhang,Shangyan Yang,Danfeng Zhang,Tao Lu,Weifang Tang

Synthesis and Biological Evaluation of 2-methoxy-N-phenyl-6-(5-phenyl-1, 3,4-oxadiazol-2-yl) pyridin-3-amine Derivatives as Antimicrobial Agents

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 4 Year: 2016 Page: 249-254
Author(s): Vasu Namani,B. Bharath Kumar Goud,Y. Bharathi Kumari,Ramesh Kumbham

Research Article

Using the Sonogashira Reaction for Preparing a New Fragment Library based on the 3-alkynylimidazo[1,2-a]pyridine Scaffold

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 7 Year: 2016 Page: 519-525
Author(s): Caroline Castera-Ducros, Hussein El-Kashef, Melanie Piednoel, Vincent Remusat, Jean-Claude Teulade, Pierre Verhaeghe, Pascal Rathelot, Patrice Vanelle

Synthesis and Crystal Structures of Some Pyridyl Aminothiazole and Thiazolidin-2-ylidene Benzamide Derivatives

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 4 Year: 2016 Page: 263-271
Author(s): Reza Heydari,Fahimeh Shahrekipour,Claudia Graiff

Research Article

A Facile Anti-selective Synthesis of 3-Nitropyridin-2-ones Using Morita- Baylis Hillman Adduct of Nitroalkene

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 8 Year: 2016 Page: 547-553
Author(s): Vijai K. Rai,Ganeshwar P. Sahu,Manorama Singh,Ankita Rai

Synthesis of Metronidazole Derivatives Containing Pyridine Ring and Anticancer Activity

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 4 Year: 2016 Page: 283-288
Author(s): Jianping Yong,Canzhong Lu,Xiaoyuan Wu

Review Article

Triggering PIK3CA Mutations in PI3K/Akt/mTOR Axis: Exploration of Newer Inhibitors and Rational Preventive Strategies

Journal: Current Pharmaceutical Design
Volume: 22 Issue: 39 Year: 2016 Page: 6039-6054
Author(s): Vivek Asati,Sanjay K. Bharti,Debarshi Kar Mahapatra,Vikas Asati,Ashok K. Budhwani

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