Search Result "1H-1"


Synthesis and Anticonvulsant Activity of Novel 3-(2-(4H-1,2,4-triazol-4- yl)ethyl)-1-alkyl-1H-indole Derivatives

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 8 Year: 2016 Page: 833-839
Author(s): Chuan-Feng Liu, Hong-Jian Zhang, Zhe-Shan Quan

Research Article

Synthesis and Antitubercular Evaluation on Novel 1-Ethyl-5-(hetero)aryl- 1,6-dihydropyrazine-2,3-dicarbonitriles and 3-Cyano-1-ethyl-5-(hetero) aryl-2(1H)-pyrazinones

Journal: Anti-Infective Agents
Volume: 14 Issue: 2 Year: 2016 Page: 139-144
Author(s): Marionella A. Kravchenko, Egor V. Verbitskiy, Sergey N. Skornyakov, Pavel A. Slepukhin, Gennagy L. Rusinov, Oleg N. Chupakhin, Valery N. Charushin

Research Article

Ionic Liquid: An Efficient and Facile Catalyst for the Synthesis of Trisubstituted Imidazole Derivatives via Multi-Component Pathway Using Green Techniques

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 10 Year: 2016 Page: 742-748
Author(s): Gopinath D. Shirole,Sharad N. Shelke

Research Article

An Efficient and Rapid Microwave-Assisted Synthesis of 1-acetyl-1Hindol- 3-yl Acetates

Journal: Current Microwave Chemistry
Volume: 3 Issue: 3 Year: 2016 Page: 247-257
Author(s): Jay P. Parshotam,John A. Brazier,Richard Bovill,Helen M.I. Osborn

Rational Design, Synthesis, Anti-HIV-1 RT and Anti-microbial Activity of Novel 2-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)-N-phenylpropanamide Derivatives

Journal: Anti-Infective Agents
Volume: 14 Issue: 1 Year: 2016 Page: 63-73
Author(s): Subhash Chander,Penta Ashok,Rajnish P. Singh,Prabhat N. Jha,Yong-Tang Zheng,Ping Wang,Sankaranarayanan Murugesan

New N,N,N’,N’-tetradentate Pyrazoly Agents: Synthesis and Evaluation of their Antifungal and Antibacterial Activities

Journal: Medicinal Chemistry
Volume: 12 Issue: 1 Year: 2016 Page: 83-89
Author(s): Farid Abrigach,Btissam Bouchal,Olivier Riant,Yohan Mace,Abdelilah Takfaoui,Smaail Radi,Abdelouahad Oussaid,Mohammed Bellaoui,Rachid Touzani

A Series of 2,4(1H,3H)-Quinazolinedione Derivatives: Synthesis and Biological Evaluation as Potential Anticancer Agents

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 1 Year: 2016 Page: 64-76
Author(s): Hulya Akgun,Demet Us Yilmaz,Rengul Cetin Atalay,Damla Gozen

Synthesis and Evaluation of Anticonvulsant Activities of Pyrazol yl Semicarbazones. Part II

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 8 Year: 2016 Page: 800-808
Author(s): Ming-Xia Song, Yi Wu, Xian-Qing Deng

Research Article

Quaternary Ammonium Ionic Liquid as a Dual Solvent-Catalyst in Biginelli Reaction

Journal: Letters in Organic Chemistry
Volume: 13 Issue: 7 Year: 2016 Page: 526-530
Author(s): Imane Tebabel, Taoues Boumoud, Boudjemaa Boumoud, Debache Abdelmadjid

Antimicrobial and Anti-biofilm Activity of Thiourea Derivatives Bearing 3-amino-1H-1,2,4-triazole Scaffold

Journal: Medicinal Chemistry
Volume: 12 Issue: 5 Year: 2016 Page: 478-488
Author(s): Joanna Stefanska,Karolina Stepien,Anna Bielenica,Daniel Szulczyk,Barbara Miroslaw,Anna E Koziol,Giuseppina Sanna,Filippo Iuliano,Silvia Madeddu,Michal Jozwiak,Marta Struga

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